SCHEMBL6585747

SCHEMBL6585747

O=C(Cl)c1ccc(F)c(CC(F)(F)F)c1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MRGPRX4 Q96LA9 1/20 0.38
CES2 O00748 2/20 0.37
CES1 P23141 2/20 0.37
KCNQ3 O43525 4/20 0.33
KCNQ2 O43526 4/20 0.33
KCNE1 P15382 4/20 0.33
KCNQ1 P51787 4/20 0.33
ALDH1A1 P00352 3/20 0.32
ALOX15 P16050 1/20 0.32
PLOD2 O00469 1/20 0.32
TRPV1 Q8NER1 1/20 0.31
RIPK1 Q13546 1/20 0.31
KIF11 P52732 1/20 0.31
EPHX2 P34913 1/20 0.31
NR1H4 Q96RI1 1/20 0.31
TSHR P16473 1/20 0.31
CHRNA1 P02708 1/20 0.30
CHRNG P07510 1/20 0.30
CHRNB1 P11230 1/20 0.30
CHRNB2 P17787 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7738818 0.84 ALDH1A1 (0.32) CES2CES1ALDH1A1EPHX2NR1H4
SCHEMBL27527292 0.84 MRGPRX4 (0.48) MRGPRX4CES2CES1ALDH1A1EPHX2
SCHEMBL31435271 0.80 CES2 (0.41) MRGPRX4CES2CES1ALDH1A1ALOX15
SCHEMBL4123543 0.80 CES2 (0.41) MRGPRX4CES2CES1ALDH1A1ALOX15
SCHEMBL5591797 0.79 CES2 (0.39) MRGPRX4CES2CES1KCNQ3KCNQ2
SCHEMBL20256821 0.74 MPO (0.40) ALDH1A1ALOX15
SCHEMBL11669995 0.74 ALDH1A1 (0.54) CES2CES1KCNQ3KCNQ2KCNE1
SCHEMBL192962 0.73 CES2 (0.67) CES2CES1KCNQ3KCNQ2KCNE1
SCHEMBL29470947 0.73 CES2 (0.67) CES2CES1KCNQ3KCNQ2KCNE1
SCHEMBL759728 0.73 KCNQ3 (0.54) CES2CES1KCNQ3KCNQ2KCNE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1379506-A2 SUBSTITUTED CARBOXAMIDES ELI LILLY AND COMPANY (US) 2004-01-14 EP disclosed
WO-2002064567-A2 SUBSTITUTED CARBOXAMIDES AS INHIBITORS OF FACTOR XA ELI LILLY AND COMPANY (US) 2002-08-22 WO disclosed