SCHEMBL6586196

SCHEMBL6586196

CN1CCN(c2ccncc2-c2nc3c(OC(N)=O)cccc3[nH]2)CC1

nearest known ligand 0.44

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 1/20 0.44
PRKCZ Q05513 9/20 0.42
PARP1 P09874 6/20 0.41
CDK2 P24941 8/20 0.41
WNT1 P04628 3/20 0.40
TGFBR1 P36897 2/20 0.40
HTR6 P50406 1/20 0.39
PARP2 Q9UGN5 3/20 0.39
CDK4 P11802 1/20 0.39
CCNA2 P20248 1/20 0.39
CCND1 P24385 1/20 0.39
CCND3 P30281 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6589131 0.90 AURKB (0.40) PRKCZPARP1PARP2
SCHEMBL6590870 0.89 AURKB (0.51) PARP1
SCHEMBL6587212 0.86 AURKA (0.50) PARP1
SCHEMBL6805985 0.85 PARP1 (0.56) PRKCZPARP1PARP2
SCHEMBL6583719 0.83 PARP1 (0.43) PARP1
SCHEMBL6587697 0.82 AURKB (0.44) PARP1
SCHEMBL6587758 0.80 PARP1 (0.57) PRKCZPARP1PARP2
SCHEMBL6587920 0.80 PARP1 (0.46) PRKCZPARP1PARP2
SCHEMBL6581295 0.79 AURKB (0.56) PRKCZPARP1PARP2
SCHEMBL6874969 0.78 PARP1 (0.51) PARP1HTR6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1177178-B1 HETEROCYCLICALLY SUBSTITUTED BENZIMIDAZOLES, THE PRODUCTION AND APPLICATION THEREOF ABBOTT GMBH & CO KG (DE) 2004-12-29 EP disclosed