SCHEMBL6589131

SCHEMBL6589131

CCN1CCN(c2ccncc2-c2nc3c(OC(N)=O)cccc3[nH]2)CC1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AURKB Q96GD4 4/20 0.40
AURKA O14965 3/20 0.40
PARP1 P09874 6/20 0.39
PARP2 Q9UGN5 1/20 0.39
GNRHR P30968 6/20 0.38
SMN1; SMN2 Q16637 1/20 0.37
KDR P35968 1/20 0.37
HTR2A P28223 1/20 0.36
PKN1 Q16512 2/20 0.36
PKN2 Q16513 2/20 0.36
SSTR5 P35346 1/20 0.36
PLK4 O00444 1/20 0.36
MAPK13 O15264 1/20 0.36
DYRK3 O43781 1/20 0.36
ROCK2 O75116 1/20 0.36
RPS6KA5 O75582 1/20 0.36
PRKD3 O94806 1/20 0.36
MAP4K4 O95819 1/20 0.36
CHEK2 O96017 1/20 0.36
PIM1 P11309 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6590870 0.91 AURKB (0.51) AURKBAURKAPARP1GNRHRKDR
SCHEMBL6586196 0.90 BRD4 (0.44) PARP1PARP2PRKCZ
SCHEMBL6587212 0.89 AURKA (0.50) AURKBAURKAPARP1GNRHRKDR
SCHEMBL6810101 0.86 AURKB (0.54) AURKBAURKAPARP1PARP2KDR
SCHEMBL6580718 0.81 AURKB (0.61) AURKBAURKAPARP1GNRHRKDR
SCHEMBL6588603 0.79 AURKA (0.63) AURKBAURKAPARP1GNRHRKDR
SCHEMBL6583719 0.79 PARP1 (0.43) AURKBAURKAPARP1GNRHRKDR
SCHEMBL6587697 0.78 AURKB (0.44) AURKBAURKAPARP1KDRPRKD3
SCHEMBL6801983 0.78 AURKB (0.68) AURKBAURKAPARP1PARP2KDR
SCHEMBL6587758 0.78 PARP1 (0.57) AURKBAURKAPARP1PARP2SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1177178-B1 HETEROCYCLICALLY SUBSTITUTED BENZIMIDAZOLES, THE PRODUCTION AND APPLICATION THEREOF ABBOTT GMBH & CO KG (DE) 2004-12-29 EP disclosed
EP-1177178-A1 HETEROCYCLICALLY SUBSTITUTED BENZIMIDAZOLES, THE PRODUCTION AND APPLICATION THEREOF BASF AKTIENGESELLSCHAFT (DE) 2002-02-06 EP disclosed
WO-2000068206-A1 HETEROCYCLICALLY SUBSTITUTED BENZIMIDAZOLES, THE PRODUCTION AND APPLICATION THEREOF BASF AKTIENGESELLSCHAFT (DE) 2000-11-16 WO disclosed