SCHEMBL6587971

SCHEMBL6587971

NC(=O)Oc1cccc2[nH]c(-c3cnc4ccccc4n3)nc12

nearest known ligand 0.59

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 11/20 0.59
ADORA1 P30542 7/20 0.59
ADORA2A P29274 4/20 0.59
CBFB Q13951 2/20 0.44
ALDH1A1 P00352 1/20 0.44
TP53 P04637 1/20 0.44
CYP3A4 P08684 1/20 0.44
CYP2D6 P10635 1/20 0.44
HPGD P15428 1/20 0.44
ALOX15 P16050 1/20 0.44
CYP2C19 P33261 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
HSD17B10 Q99714 1/20 0.44
PARP1 P09874 5/20 0.43
HPSE Q9Y251 1/20 0.41
DHODH Q02127 3/20 0.40
PARP2 Q9UGN5 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6585381 0.82 CBFB (0.67) CBFBALDH1A1TP53CYP3A4CYP2D6
SCHEMBL6806558 0.82 ADORA3 (0.63) ADORA3ADORA1ADORA2APARP1DHODH
SCHEMBL6590890 0.80 METAP2 (0.50) CBFBALDH1A1TP53CYP3A4CYP2D6
SCHEMBL6585540 0.77 CBFB (0.47) CBFBALDH1A1TP53CYP3A4CYP2D6
SCHEMBL6585207 0.76 PARP1 (0.51) CBFBALDH1A1TP53CYP3A4CYP2D6
SCHEMBL31061052 0.75 ADORA3 (1.00) ADORA3ADORA1ADORA2ACBFBALDH1A1
SCHEMBL31060640 0.75 ADORA3 (1.00) ADORA3ADORA1ADORA2ACBFB
SCHEMBL6589950 0.75 PKN1 (0.46) ALOX15PARP1HPSEDHODHPARP2
SCHEMBL6590709 0.74 PKN1 (0.66) ALOX15PARP1HPSEDHODHPARP2
SCHEMBL6590776 0.74 PARP1 (0.46) CBFBALDH1A1TP53CYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1177178-B1 HETEROCYCLICALLY SUBSTITUTED BENZIMIDAZOLES, THE PRODUCTION AND APPLICATION THEREOF ABBOTT GMBH & CO KG (DE) 2004-12-29 EP disclosed
EP-1177178-A1 HETEROCYCLICALLY SUBSTITUTED BENZIMIDAZOLES, THE PRODUCTION AND APPLICATION THEREOF BASF AKTIENGESELLSCHAFT (DE) 2002-02-06 EP disclosed
WO-2000068206-A1 HETEROCYCLICALLY SUBSTITUTED BENZIMIDAZOLES, THE PRODUCTION AND APPLICATION THEREOF BASF AKTIENGESELLSCHAFT (DE) 2000-11-16 WO disclosed