SCHEMBL6589560

SCHEMBL6589560

COc1cc2c(cc1F)SC(C)(C)CC2=O

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.47
KDM4E B2RXH2 5/20 0.47
HPGD P15428 1/20 0.47
KLK7 P49862 1/20 0.47
CA1 P00915 1/20 0.34
CA2 P00918 1/20 0.34
CA7 P43166 1/20 0.34
CA9 Q16790 1/20 0.34
NCOA1 Q15788 1/20 0.34
NCOA3 Q9Y6Q9 1/20 0.34
TDP2 O95551 1/20 0.34
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
TUBB4A P04350 1/20 0.32
TUBB P07437 1/20 0.32
TUBA3C P0DPH7 1/20 0.32
TUBA1B P68363 1/20 0.32
TUBA4A P68366 1/20 0.32
TUBB4B P68371 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6592551 0.80 ALDH1A1 (0.33) ALDH1A1KDM4EHPGDKLK7MEN1
SCHEMBL31260280 0.72 ALDH1A1 (0.57) ALDH1A1KDM4EKLK7CA1CA2
SCHEMBL1140756 0.72 ALDH1A1 (0.47) ALDH1A1KDM4EKLK7CA1CA2
SCHEMBL1987343 0.72 ALDH1A1 (0.57) ALDH1A1KDM4EKLK7CA1CA2
SCHEMBL31260278 0.72 ALDH1A1 (0.57) ALDH1A1KDM4EKLK7CA1CA2
SCHEMBL68563 0.68 KDM4E (0.48) ALDH1A1KDM4EHPGDCA1CA2
SCHEMBL68066 0.67 VHL (0.50) ALDH1A1KDM4EHPGDMEN1KMT2A
SCHEMBL9379290 0.67 PGR (0.42) ALDH1A1KDM4EHPGDMEN1KMT2A
SCHEMBL12471284 0.67 MEN1 (0.47) ALDH1A1KDM4EHPGDNCOA1TDP2
SCHEMBL606742 0.66 PTGS2 (0.47) ALDH1A1KDM4EHPGDMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1042313-B1 BENZOPYRAN AND BENZOTHIOPYRAN DERIVATIVES HAVING RETINOID ANTAGONIST LIKE ACTIVITY ALLERGAN INC (US) 2004-04-28 EP disclosed
EP-1042313-A1 BENZOPYRAN AND BENZOTHIOPYRAN DERIVATIVES HAVING RETINOID ANTAGONIST LIKE ACTIVITY Allergan Sales, Inc. (US) 2000-10-11 EP disclosed
US-5958954-A 2,2-DIALKYL-4-ARYL-SUBSTITUTED BENZOPYRAN AND BENZOTHIOPYRAN DERIVATIVES ALLERGAN SALES, INC. (US) 1999-09-28 US disclosed
WO-1999033821-A1 BENZOPYRAN AND BENZOTHIOPYRAN DERIVATIVES HAVING RETINOID ANTAGONIST-LIKE ACTIVITY ALLERGAN SALES, INC. (US) 1999-07-08 WO disclosed