SCHEMBL6589849

SCHEMBL6589849

O=C(NCc1nc(Cl)ccc1OC[C@@H]1CCCCN1)c1cccnc1

nearest known ligand 0.44

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.42
CHRNA3 P32297 4/20 0.40
CHRNB4 P30926 2/20 0.40
NPC1 O15118 1/20 0.40
CHRNB2 P17787 1/20 0.40
CHRNA4 P43681 1/20 0.40
THRB P10828 1/20 0.40
MAPT P10636 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6584722 0.79 NPC1 (0.42) TSHRCHRNA3NPC1
SCHEMBL13100535 0.72 THRB (0.54) NPC1THRBMAPT
SCHEMBL13100536 0.68 LMNA (0.49) CHRNA3CHRNB4CHRNB2CHRNA4MAPT
SCHEMBL24154367 0.67 CHRNA3 (0.78) CHRNA3CHRNB4CHRNB2CHRNA4
SCHEMBL1648049 0.65 TSHR (0.63) TSHRCHRNA3CHRNB4CHRNB2CHRNA4
Hydrochloric Acid SCHEMBL30983201 0.65 CHRNA3 (0.56) CHRNA3CHRNB4CHRNB2CHRNA4
SCHEMBL905201 0.64 CHRNA3 (0.81) CHRNA3CHRNB4CHRNB2CHRNA4
SCHEMBL905236 0.64 CHRNA3 (0.81) CHRNA3CHRNB4CHRNB2CHRNA4
SCHEMBL3942452 0.64 CHRNA3 (0.81) CHRNA3CHRNB4CHRNB2CHRNA4
Hydrochloric Acid SCHEMBL7840031 0.63 CHRNA3 (0.78) CHRNA3CHRNB4CHRNB2CHRNA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0934308-B1 3-PYRIDYLOXYMETHYL HETEROCYCLIC ETHER COMPOUNDS USEFUL IN CONTROLLING CHEMICAL SYNAPTIC TRANSMISSION ABBOTT LAB (US) 2004-08-11 EP claimed