SCHEMBL6590774

SCHEMBL6590774

CC(C)CC(NC(=O)c1ccc(F)cc1)C(=O)N(C1CCCNC[C@@H]1O)S(=O)(=O)C1=NC=CCC1=O

nearest known ligand 0.35

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CTSL P07711 5/20 0.35
MAPK14 Q16539 2/20 0.34
CTSB P07858 3/20 0.33
CTSK P43235 2/20 0.33
CTSS P25774 1/20 0.33
CA1 P00915 3/20 0.33
CA12 O43570 2/20 0.33
CA9 Q16790 2/20 0.33
USP30 Q70CQ3 1/20 0.32
CA2 P00918 2/20 0.32
CNR2 P34972 3/20 0.31
CNR1 P21554 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6593138 0.89 CTSL (0.31) CTSLCTSBCTSKCTSS
SCHEMBL7386818 0.88
SCHEMBL4763320 0.87 CTSL (0.37) CTSLMAPK14CTSBCTSKCTSS
SCHEMBL6896141 0.84 MAPK1 (0.32) CTSLCTSBCTSKCTSS
SCHEMBL4765376 0.76 CTSK (0.31) CTSLCTSBCTSKCTSS
SCHEMBL6211401 0.76 CTSK (0.37) CTSLCTSBCTSKCTSS
SCHEMBL6590804 0.75 CTSL (0.31) CTSLCTSKCTSS
SCHEMBL4767192 0.75 TAS1R3 (0.44)
SCHEMBL6589335 0.75
SCHEMBL4766715 0.74 CTSK (0.37) CTSLCTSBCTSKCTSS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1307204-A4 PROTEASE INHIBITORS SMITHKLINE BEECHAM CORP (US) 2004-06-02 EP disclosed
EP-1307204-A1 PROTEASE INHIBITORS SmithKline Beecham Corporation (US) 2003-05-07 EP disclosed
WO-2001095911-A1 PROTEASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2001-12-20 WO disclosed