SCHEMBL6593140

SCHEMBL6593140

N#Cc1cccc2c(OCc3ccccc3)c(C#Cc3ccccc3)c(C(=O)O)nc12

nearest known ligand 0.38

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
XDH P47989 3/20 0.38
PPIA P62937 1/20 0.37
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36
MCL1 Q07820 1/20 0.36
FFAR1 O14842 1/20 0.36
AKR1B1 P15121 1/20 0.36
ADORA3 P0DMS8 1/20 0.35
PTPN1 P18031 1/20 0.35
PTPN6 P29350 1/20 0.35
PTPN11 Q06124 1/20 0.35
MAOB P27338 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6080436 0.91 ADORA3 (0.41) XDHPPIAFFAR1AKR1B1ADORA3
Benzene SCHEMBL6592619 0.88 XDH (0.39) XDHKDM4EALDH1A1MAOB
SCHEMBL6593145 0.83 XDH (0.40) XDHMCL1FFAR1
SCHEMBL6594157 0.83 XDH (0.40) XDHKDM4EALDH1A1MAOB
SCHEMBL6080444 0.82 XDH (0.38) XDHPPIAKDM4EADORA3MAOB
SCHEMBL6079768 0.81 ALDH1A1 (0.38) KDM4EALDH1A1MCL1FFAR1ADORA3
SCHEMBL6080295 0.80 KDM4A (0.38) KDM4EALDH1A1MCL1PTPN1PTPN6
SCHEMBL6079492 0.78 XDH (0.41) XDHADORA3MAOB
SCHEMBL6080478 0.76 XDH (0.39) XDHKDM4EALDH1A1MAOB
SCHEMBL6080232 0.73 PTGER1 (0.43) PPIAADORA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1451159-A1 COMPOSITIONS DERIVED FROM QUINOLINE AND QUINOXALINE, PREPARATION AND USE THEREOF NEURO3D (FR) 2004-09-01 EP claimed
WO-2003010146-A1 COMPOSITIONS DERIVED FROM QUINOLINE AND QUINOXALINE, PREPARATION AND USE THEREOF NEURO3D (FR) 2003-02-06 WO claimed
EP-1451159-A1 COMPOSITIONS DERIVED FROM QUINOLINE AND QUINOXALINE, PREPARATION AND USE THEREOF NEURO3D (FR) 2004-09-01 EP disclosed
WO-2003010146-A1 COMPOSITIONS DERIVED FROM QUINOLINE AND QUINOXALINE, PREPARATION AND USE THEREOF NEURO3D (FR) 2003-02-06 WO disclosed