SCHEMBL6594338

SCHEMBL6594338

O=C(O)c1nc2c([N+](=O)[O-])cccc2c(O)c1Br

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.46
MEN1 O00255 5/20 0.46
KMT2A Q03164 5/20 0.46
KDM4E B2RXH2 3/20 0.46
MAPT P10636 3/20 0.46
TSHR P16473 2/20 0.46
CYP2D6 P10635 2/20 0.46
CYP2C19 P33261 2/20 0.46
CYP1A2 P05177 1/20 0.46
CYP3A4 P08684 1/20 0.46
ALOX15 P16050 1/20 0.46
MAPK1 P28482 1/20 0.46
NOS1 P29475 1/20 0.46
NOS2 P35228 1/20 0.46
BLM P54132 1/20 0.46
GPR35 Q9HC97 2/20 0.44
TDP1 Q9NUW8 3/20 0.41
PDE10A Q9Y233 1/20 0.40
CTSB P07858 1/20 0.40
GAA P10253 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6594345 1.00 ALDH1A1 (0.46) ALDH1A1MEN1KMT2AKDM4EMAPT
SCHEMBL6080451 0.86 ALDH1A1 (0.43) ALDH1A1MEN1KMT2AKDM4EMAPT
SCHEMBL6080679 0.84 TSHR (0.49) ALDH1A1MEN1KMT2AKDM4EMAPT
SCHEMBL6080329 0.81 KMT2A (0.42) ALDH1A1MEN1KMT2AKDM4EMAPT
SCHEMBL6079406 0.81 GPR35 (0.41) ALDH1A1MEN1KMT2AKDM4EMAPT
SCHEMBL6080956 0.81 FBP1 (0.51) ALDH1A1MEN1KMT2AKDM4EMAPT
SCHEMBL6079956 0.80 KDM4E (0.44) ALDH1A1KMT2AKDM4ECYP2D6CYP2C19
SCHEMBL6594653 0.78 ALDH1A1 (0.38) ALDH1A1MEN1KMT2AKDM4EMAPT
SCHEMBL6594657 0.78 ALDH1A1 (0.38) ALDH1A1MEN1KMT2AKDM4EMAPT
SCHEMBL6079987 0.77 MMP2 (0.41) ALDH1A1MEN1KMT2AKDM4EMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1451159-A1 COMPOSITIONS DERIVED FROM QUINOLINE AND QUINOXALINE, PREPARATION AND USE THEREOF NEURO3D (FR) 2004-09-01 EP claimed
WO-2003010146-A1 COMPOSITIONS DERIVED FROM QUINOLINE AND QUINOXALINE, PREPARATION AND USE THEREOF NEURO3D (FR) 2003-02-06 WO claimed
EP-1451159-A1 COMPOSITIONS DERIVED FROM QUINOLINE AND QUINOXALINE, PREPARATION AND USE THEREOF NEURO3D (FR) 2004-09-01 EP disclosed
WO-2003010146-A1 COMPOSITIONS DERIVED FROM QUINOLINE AND QUINOXALINE, PREPARATION AND USE THEREOF NEURO3D (FR) 2003-02-06 WO disclosed