SCHEMBL6595415

SCHEMBL6595415

CC1CC(c2cccc3sccc23)=CCN1

nearest known ligand 0.40

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ADRA2A P08913 1/20 0.40
ADRA2B P18089 1/20 0.40
SLC6A2 P23975 1/20 0.33
SLC6A4 P31645 1/20 0.33
SLC6A3 Q01959 1/20 0.33
GSK3A P49840 1/20 0.33
GSK3B P49841 1/20 0.33
HTR1A P08908 1/20 0.32
DRD2 P14416 1/20 0.32
HTR2A P28223 1/20 0.32
ATR Q13535 1/20 0.31
ATRIP Q8WXE1 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6594982 0.74 HTR2C (0.47) ADRA2AADRA2BDRD2
SCHEMBL5153625 0.70 ADRA2A (0.56) ADRA2AADRA2BSLC6A2SLC6A4SLC6A3
SCHEMBL4790016 0.69 CYP2A6 (0.35) HTR1A
SCHEMBL4789469 0.69 ALDH1A1 (0.35) ADRA2AADRA2BHTR2A
SCHEMBL4788776 0.69 IDH1 (0.36) HTR1A
Hydrochloric Acid SCHEMBL7766719 0.69 HTR7 (0.36)
SCHEMBL4605690 0.69 ALDH1A1 (0.40) HTR2A
SCHEMBL4790431 0.69 PBRM1 (0.41)
Hydrochloric Acid SCHEMBL6336129 0.68
SCHEMBL22053914 0.67 DRD2 (0.45) HTR1ADRD2HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1204660-B1 SEROTONERGIC BENZOTHIOPHENES LILLY CO ELI (US) 2004-10-20 EP disclosed
EP-1204660-A1 SEROTONERGIC BENZOTHIOPHENES ELI LILLY AND COMPANY (US) 2002-05-15 EP disclosed
WO-2001009126-A1 SEROTONERGIC BENZOTHIOPHENES ELI LILLY AND COMPANY (US) 2001-02-08 WO disclosed