SCHEMBL6596226

SCHEMBL6596226

CC=C(C(=O)ON=[N+]=[N-])c1ccccc1OCc1ccccc1

nearest known ligand 0.46

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HTT P42858 2/20 0.46
SGMS2 Q8NHU3 3/20 0.45
NPC1 O15118 2/20 0.43
RXRA P19793 1/20 0.43
PARP1 P09874 1/20 0.43
GAA P10253 1/20 0.43
ATM Q13315 1/20 0.42
KDM4E B2RXH2 2/20 0.42
POLB P06746 2/20 0.42
MAPT P10636 2/20 0.42
RECQL P46063 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
PTGER1 P34995 1/20 0.42
MEN1 O00255 3/20 0.42
KMT2A Q03164 3/20 0.42
LIPE Q05469 1/20 0.42
L3MBTL1 Q9Y468 2/20 0.41
ALDH1A1 P00352 2/20 0.41
LMNA P02545 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1097809 0.81 SGMS2 (0.59) HTTSGMS2NPC1GAAMAPT
SCHEMBL9642440 0.81 SGMS2 (0.59) HTTSGMS2NPC1GAAMAPT
SCHEMBL8827709 0.79 SGMS2 (0.56) HTTSGMS2NPC1PARP1GAA
SCHEMBL9731418 0.79 SGMS2 (0.50) HTTSGMS2NPC1PARP1GAA
SCHEMBL6938166 0.72 SGMS2 (0.58) HTTSGMS2NPC1GAAMAPT
SCHEMBL10443318 0.72 SGMS2 (0.58) HTTSGMS2NPC1GAAMAPT
SCHEMBL9231981 0.71 SGMS2 (0.54) HTTSGMS2NPC1PARP1GAA
SCHEMBL712291 0.71 SGMS2 (0.57) HTTSGMS2NPC1GAAMAPT
SCHEMBL7164705 0.71 SGMS2 (0.57) HTTSGMS2NPC1GAAMAPT
SCHEMBL316291 0.71 SGMS2 (0.53) HTTSGMS2NPC1GAAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1150954-B1 ANTI-IMFLAMMATORY INDOLE DERIVATIVES ASTRAZENECA AB (SE) 2004-10-13 EP disclosed
US-6569888-B1 Such as ethyl-N-(dichlorobenzyl)-4-(3-hydroxypropylthio) indole-2-carboxylate; for treatment of arthritis ASTRAZENECA AB (SE) 2003-05-27 US disclosed