SCHEMBL6597293

SCHEMBL6597293

O=C(O)Oc1cnn(-c2ccccc2C(F)(F)F)c1C1CC1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KEAP1 Q14145 1/20 0.41
NFE2L2 Q16236 1/20 0.41
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
RBP4 P02753 5/20 0.38
SLC9A1 P19634 2/20 0.38
SLC9A2 Q9UBY0 2/20 0.38
SLC16A3 O15427 1/20 0.35
SLC16A1 P53985 1/20 0.35
SCN9A Q15858 1/20 0.35
NOTUM Q6P988 1/20 0.35
TTR P02766 1/20 0.35
POLB P06746 1/20 0.34
MAPT P10636 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
CYP2C9 P11712 1/20 0.34
CYP2C19 P33261 1/20 0.34
HTR2B P41595 1/20 0.34
MAPK14 Q16539 1/20 0.34
ALDH1A1 P00352 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6314631 0.82 NFE2L2 (0.64) KEAP1NFE2L2MEN1KMT2ARBP4
SCHEMBL6312965 0.76 TP53 (0.49) KEAP1NFE2L2MEN1KMT2APOLB
SCHEMBL6600754 0.75 SLC9A1 (0.42) KEAP1NFE2L2MEN1KMT2ASLC9A1
SCHEMBL4450211 0.74 SLC9A1 (0.69) KEAP1NFE2L2MEN1KMT2ASLC9A1
SCHEMBL6600449 0.74 SLC9A1 (0.61) SLC9A1SLC9A2
Hydrochloric Acid SCHEMBL6314762 0.73 SLC9A1 (0.67) KEAP1NFE2L2MEN1KMT2ASLC9A1
SCHEMBL4450205 0.73 SLC9A1 (0.48) KEAP1NFE2L2MEN1KMT2ASLC9A1
Hydrochloric Acid SCHEMBL6321496 0.73 SLC9A1 (0.66) KEAP1NFE2L2MEN1KMT2ASLC9A1
Hydrochloric Acid SCHEMBL6314755 0.73 SLC9A1 (0.48) KEAP1NFE2L2MEN1KMT2ASLC9A1
SCHEMBL7360447 0.72 KEAP1 (0.53) KEAP1NFE2L2KMT2ASLC9A1SLC9A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1056729-B1 N-[(SUBSTITUTED FIVE-MEMBERED DI- OR TRIAZA DIUNSATURATED RING)CARBONYL]GUANIDINE DERIVATIVES FOR THE TREATMENT OF ISCHEMIA PFIZER PROD INC (US) 2004-12-29 EP claimed