SCHEMBL6600754

SCHEMBL6600754

O=C(O)Oc1cnn(-c2cccc3cccnc23)c1C1CC1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC9A1 P19634 3/20 0.42
SLC9A2 Q9UBY0 2/20 0.42
OPRM1 P35372 1/20 0.42
OPRD1 P41143 1/20 0.42
OPRK1 P41145 1/20 0.42
LMNA P02545 3/20 0.40
METAP2 P50579 1/20 0.40
METAP1 P53582 1/20 0.40
HDAC6 Q9UBN7 1/20 0.40
POLB P06746 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
ALDH1A1 P00352 3/20 0.39
HSP90AA1 P07900 1/20 0.38
KEAP1 Q14145 1/20 0.38
NFE2L2 Q16236 1/20 0.38
TSHR P16473 1/20 0.37
ESR2 Q92731 1/20 0.37
USP2 O75604 1/20 0.37
HCRTR1 O43613 1/20 0.37
HCRTR2 O43614 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6600449 0.83 SLC9A1 (0.61) SLC9A1SLC9A2OPRM1OPRD1OPRK1
SCHEMBL6312945 0.83 NFE2L2 (0.57) SLC9A1SLC9A2OPRM1OPRD1OPRK1
SCHEMBL27523940 0.77 SLC9A1 (0.43) SLC9A1SLC9A2OPRM1OPRD1OPRK1
SCHEMBL6320770 0.77 TP53 (0.48) SLC9A1SLC9A2OPRM1OPRD1OPRK1
SCHEMBL4451940 0.75 SLC9A1 (0.73) SLC9A1SLC9A2OPRM1OPRD1OPRK1
SCHEMBL6597293 0.75 KEAP1 (0.41) SLC9A1SLC9A2POLBSMN1; SMN2ALDH1A1
SCHEMBL4451936 0.74 SLC9A1 (0.52) SLC9A1SLC9A2OPRM1OPRD1OPRK1
Hydrochloric Acid SCHEMBL6314615 0.74 SLC9A1 (0.74) SLC9A1SLC9A2OPRM1OPRD1OPRK1
Hydrochloric Acid SCHEMBL6314605 0.74 SLC9A1 (0.52) SLC9A1SLC9A2OPRM1OPRD1OPRK1
SCHEMBL3415803 0.70 LMNA (0.71) LMNAMETAP2METAP1HDAC6POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1056729-B1 N-[(SUBSTITUTED FIVE-MEMBERED DI- OR TRIAZA DIUNSATURATED RING)CARBONYL]GUANIDINE DERIVATIVES FOR THE TREATMENT OF ISCHEMIA PFIZER PROD INC (US) 2004-12-29 EP claimed