SCHEMBL6597298

SCHEMBL6597298

Cc1ccc2sc(-c3ccc(OCCN4CCCC4)cc3)cc2c1

nearest known ligand 0.54

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ACHE P22303 2/20 0.54
ESR1 P03372 4/20 0.51
ESR2 Q92731 4/20 0.51
HRH3 Q9Y5N1 4/20 0.50
LTA4H P09960 3/20 0.50
CHEK1 O14757 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.47
KDM4E B2RXH2 2/20 0.46
L3MBTL1 Q9Y468 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6595152 0.88 LTA4H (0.55) ESR1ESR2HRH3LTA4H
SCHEMBL6594650 0.84 LTA4H (0.60) HRH3LTA4H
SCHEMBL6593929 0.81 ESR1 (0.56) ESR1ESR2HRH3LTA4H
SCHEMBL7774143 0.79 LTA4H (0.55) ESR1ESR2HRH3LTA4HCHEK1
SCHEMBL3968157 0.79 AXL (0.58) HRH3CHEK1
SCHEMBL7447133 0.78 HRH3 (0.73) ACHEHRH3LTA4HKDM4E
SCHEMBL13032448 0.78 JAK2 (0.65)
SCHEMBL6595869 0.77 ACHE (0.50) ACHEESR1ESR2HRH3LTA4H
SCHEMBL8337754 0.76 HRH3 (0.70) HRH3LTA4HKDM4E
SCHEMBL7445580 0.76 POLB (0.54) ESR1ESR2HRH3LTA4HCHEK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0863755-B1 ANTITHROMBOTIC DIAMINES LILLY CO ELI (US) 2004-12-15 EP disclosed
US-6265575-B1 THROMBIN INHIBITORS ELI LILLY AND COMPANY 2001-07-24 US disclosed
US-6251921-B1 ADMINISTERING THROMBIN INHIBITING DIAMINE COMPOUND TO MAMMAL ELI LILLY AND COMPANY 2001-06-26 US disclosed
US-6025382-A Antithrombotic diamines ELI LILLY AND COMPANY (US) 2000-02-15 US disclosed