SCHEMBL6597552

SCHEMBL6597552

Cc1ncn(CCCOCc2ccccc2Cl)c1CCl

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 3/20 0.41
GAA P10253 3/20 0.38
ALDH1A1 P00352 3/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
MAPT P10636 3/20 0.36
TP53 P04637 1/20 0.36
THRB P10828 1/20 0.36
LMNA P02545 4/20 0.35
KDM4E B2RXH2 2/20 0.35
USP2 O75604 1/20 0.35
TSHR P16473 1/20 0.35
HSD17B10 Q99714 1/20 0.35
BRD4 O60885 1/20 0.35
IDO1 P14902 2/20 0.34
HPGD P15428 1/20 0.34
HRH3 Q9Y5N1 1/20 0.34
RAB9A P51151 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6599977 0.89 TDP1 (0.42) TDP1GAAALDH1A1CYP3A4CYP2D6
SCHEMBL6599808 0.84 MEN1 (0.40) TDP1CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL6598217 0.84 TDP1 (0.37) TDP1GAAALDH1A1CYP3A4CYP2D6
SCHEMBL6598215 0.75 TDP1 (0.35) TDP1GAAALDH1A1CYP3A4CYP2D6
SCHEMBL6599697 0.72 ATP4A (0.42) TDP1ALDH1A1CYP3A4CYP2D6CYP2C9
SCHEMBL19055306 0.68 IDO1 (0.50) TDP1ALDH1A1CYP3A4CYP2D6CYP2C9
SCHEMBL22670134 0.67 ADORA2A (0.38) ALDH1A1LMNAPOLB
SCHEMBL4058386 0.66 IDO1 (0.55) MAPTLMNAIDO1HPGDRAB9A
SCHEMBL18596661 0.66 IDO1 (0.47) ALDH1A1CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL6602229 0.65 IDO1 (0.50) CYP3A4CYP2D6CYP2C9CYP2C19TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1169320-B1 FARNESYL TRANSFERASE INHIBITORS HAVING A PYRROLE STRUCTURE AND PROCESS FOR PREPARATION THEREOF LG CHEM INVESTMENT LTD (KR) 2004-09-22 EP disclosed
US-6511978-B1 For treating cancer, restenosis, atherosclerosis or viral infections LG LIFE SCIENCES, LTD. (KR) 2003-01-28 US disclosed
EP-1169320-A4 FARNESYL TRANSFERASE INHIBITORS HAVING A PYRROLE STRUCTURE AND PROCESS FOR PREPARATION THEREOF LG CHEM INVESTMENT LTD (KR) 2002-10-30 EP disclosed
EP-1169320-A1 FARNESYL TRANSFERASE INHIBITORS HAVING A PYRROLE STRUCTURE AND PROCESS FOR PREPARATION THEREOF LG Chem Investment, Ltd. (KR) 2002-01-09 EP disclosed
WO-2000064891-A1 FARNESYL TRANSFERASE INHIBITORS HAVING A PYRROLE STRUCTURE AND PROCESS FOR PREPARATION THEREOF LG CHEM INVESTMENT LTD. (KR) 2000-11-02 WO disclosed