SCHEMBL6598976

SCHEMBL6598976

N/C(=N\c1ccc(N2CCN(C(=O)O)CC2)cc1)c1cccs1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOS1 P29475 1/20 0.56
MAPT P10636 5/20 0.55
GAA P10253 4/20 0.55
ALDH1A1 P00352 2/20 0.55
LMNA P02545 2/20 0.55
ALOX12 P18054 1/20 0.55
KDM4E B2RXH2 2/20 0.47
L3MBTL1 Q9Y468 2/20 0.47
KMT2A Q03164 2/20 0.47
POLB P06746 1/20 0.47
PKM P14618 1/20 0.47
RECQL P46063 1/20 0.47
THRB P10828 1/20 0.47
NOS3 P29474 1/20 0.46
KCNA5 P22460 1/20 0.46
MEN1 O00255 1/20 0.46
NOD1 Q9Y239 1/20 0.46
ADRA2A P08913 1/20 0.46
ADRA2B P18089 1/20 0.46
ADRA2C P18825 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6598979 1.00 NOS1 (0.56) NOS1MAPTGAAALDH1A1LMNA
SCHEMBL6600983 0.87 NOS1 (0.52) NOS1MAPTGAAALDH1A1LMNA
SCHEMBL6600980 0.87 NOS1 (0.52) NOS1MAPTGAAALDH1A1LMNA
SCHEMBL13979808 0.85 NOS3 (0.62) NOS1NOS3
SCHEMBL4328052 0.83 MAPT (0.54) NOS1MAPTGAAALDH1A1LMNA
SCHEMBL5387053 0.83 ALDH1A1 (0.49) NOS1MAPTGAAALDH1A1LMNA
SCHEMBL5387059 0.83 ALDH1A1 (0.49) NOS1MAPTGAAALDH1A1LMNA
Hydrochloric Acid SCHEMBL4310959 0.82 MAPT (0.53) NOS1MAPTGAAALDH1A1LMNA
SCHEMBL6602083 0.82 NOS3 (0.49) NOS1NOS3
SCHEMBL6602079 0.82 NOS3 (0.49) NOS1NOS3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1265891-B1 NOVEL LIPOIC ACID HETEROCYCLIC OR BENZENE DERIVATIVES, PREPARATION AND USE THEREOF AS MEDICINES CONSEILS DE RECH SET D APPLIC (FR) 2004-12-29 EP disclosed
EP-1265891-A2 NOVEL LIPOIC ACID HETEROCYCLIC OR BENZENE DERIVATIVES, PREPARATION AND USE THEREOF AS MEDICINES SOCIETE DE CONSEILS DE RECHERCHES ET D'APPLICATIONS SCIENTIFIQUES (S.C.R.A.S.) (FR) 2002-12-18 EP disclosed
WO-2001068643-A2 NOVEL LIPOIC ACID HETEROCYCLIC OR BENZENE DERIVATIVES, PREPARATION AND USE THEREOF AS MEDICINES SOCIETE DE CONSEILS DE RECHERCHES ET D'APPLICATIONS SCIENTIFIQUES (S.C.R.A.S.) (FR) 2001-09-20 WO disclosed