SCHEMBL6599168

SCHEMBL6599168

Cc1ccc2scc(CC(=O)CCl)c2c1

nearest known ligand 0.51

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
KEAP1 Q14145 1/20 0.51
NFE2L2 Q16236 1/20 0.51
CA2 P00918 1/20 0.50
TP53 P04637 4/20 0.45
SMN1; SMN2 Q16637 2/20 0.45
RXFP1 Q9HBX9 1/20 0.45
UTS2R Q9UKP6 1/20 0.42
MTNR1A P48039 7/20 0.42
MTNR1B P49286 3/20 0.42
CYP2A6 P11509 1/20 0.39
LMNA P02545 1/20 0.38
RAB9A P51151 1/20 0.38
MAPT P10636 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2251923 0.84 KEAP1 (0.73) KEAP1NFE2L2CA2SMN1; SMN2UTS2R
SCHEMBL1520186 0.83 KEAP1 (0.68) KEAP1NFE2L2CA2TP53SMN1; SMN2
SCHEMBL9751552 0.82 CA2 (0.56) KEAP1NFE2L2CA2TP53SMN1; SMN2
SCHEMBL9314600 0.79 CA2 (0.53) KEAP1NFE2L2CA2TP53SMN1; SMN2
SCHEMBL5179133 0.79 CA2 (0.55) KEAP1NFE2L2CA2TP53SMN1; SMN2
SCHEMBL2248697 0.78 CYP2A6 (0.58) KEAP1NFE2L2CA2TP53SMN1; SMN2
SCHEMBL19627156 0.78 CA2 (0.49) KEAP1NFE2L2CA2TP53SMN1; SMN2
SCHEMBL10266973 0.77 CA2 (0.60) KEAP1NFE2L2CA2TP53MTNR1A
SCHEMBL5267734 0.76 CYP2A6 (0.58) KEAP1NFE2L2CA2TP53SMN1; SMN2
SCHEMBL5267998 0.76 LMNA (0.54) KEAP1NFE2L2CA2TP53LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1337528-B1 BENZOTHIOPHENE DERIVATIVE COMPOUNDS, PROCESS OF PREPARATION AND USE THEREOF VITA LAB (ES) 2004-08-04 EP disclosed