SCHEMBL9751552

SCHEMBL9751552

Cc1ccc2scc(CC(N)=O)c2c1

nearest known ligand 0.56

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CA2 P00918 1/20 0.56
KEAP1 Q14145 1/20 0.50
NFE2L2 Q16236 1/20 0.50
TP53 P04637 4/20 0.47
SMN1; SMN2 Q16637 2/20 0.47
RXFP1 Q9HBX9 1/20 0.47
UTS2R Q9UKP6 1/20 0.43
ICMT O60725 2/20 0.42
ALDH1A1 P00352 1/20 0.41
RAB9A P51151 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
MTNR1A P48039 3/20 0.41
MTNR1B P49286 2/20 0.41
CYP2A6 P11509 2/20 0.41
MAPT P10636 3/20 0.40
USP2 O75604 1/20 0.39
THRB P10828 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1520186 0.86 KEAP1 (0.68) CA2KEAP1NFE2L2TP53SMN1; SMN2
SCHEMBL8020393 0.85 CA2 (0.53) CA2KEAP1NFE2L2TP53SMN1; SMN2
SCHEMBL6599168 0.82 KEAP1 (0.51) CA2KEAP1NFE2L2TP53SMN1; SMN2
SCHEMBL9314600 0.82 CA2 (0.53) CA2KEAP1NFE2L2TP53SMN1; SMN2
SCHEMBL8605628 0.82 MTNR1A (0.59) CA2KEAP1NFE2L2TP53SMN1; SMN2
SCHEMBL28564709 0.81 MTNR1A (0.57) CA2KEAP1NFE2L2TP53SMN1; SMN2
SCHEMBL31164712 0.81 MTNR1A (0.57) CA2KEAP1NFE2L2TP53SMN1; SMN2
SCHEMBL6202916 0.81 KEAP1 (0.75) CA2KEAP1NFE2L2SMN1; SMN2UTS2R
SCHEMBL28563290 0.81 CYP2A6 (0.64) CA2KEAP1NFE2L2TP53UTS2R
SCHEMBL19627156 0.81 CA2 (0.49) CA2KEAP1NFE2L2TP53SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0422119-A4 BENZOTHIOPHENE DERIVATIVES USEFUL FOR MODIFYING FEEDING BEHAVIOR AND OBSESSIVE-COMPULSIVE BEHAVIOR 1991-11-13 EP disclosed
EP-0422119-A1 BENZOTHIOPHENE DERIVATIVES USEFUL FOR MODIFYING FEEDING BEHAVIOR AND OBSESSIVE-COMPULSIVE BEHAVIOR NEUREX CORPORATION (US) 1991-04-17 EP disclosed
WO-1989012447-A1 BENZOTHIOPHENE DERIVATIVES USEFUL FOR MODIFYING FEEDING BEHAVIOR AND OBSESSIVE-COMPULSIVE BEHAVIOR NEUREX CORPORATION (US) 1989-12-28 WO disclosed