SCHEMBL6599683

SCHEMBL6599683

c1ccc(NCCc2c[nH]c3ccccc23)cc1

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 3/20 0.71
HTR1A P08908 2/20 0.71
HTR6 P50406 2/20 0.71
DRD2 P14416 1/20 0.71
HTR7 P34969 1/20 0.71
KMT2A Q03164 6/20 0.67
POLB P06746 1/20 0.67
SLC2A1 P11166 1/20 0.67
RAD52 P43351 1/20 0.67
ALDH1A1 P00352 2/20 0.66
KDM4E B2RXH2 1/20 0.66
HTT P42858 1/20 0.66
HRH3 Q9Y5N1 4/20 0.65
MC5R P33032 1/20 0.64
MC3R P41968 1/20 0.64
MC1R Q01726 1/20 0.64
MEN1 O00255 5/20 0.63
SMN1; SMN2 Q16637 2/20 0.62
MAPT P10636 1/20 0.62
G6PD P11413 1/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL11602872 0.98 HTR2A (0.70) HTR2AHTR1AHTR6DRD2HTR7
Oxalic Acid SCHEMBL6603520 0.93 KMT2A (0.67) HTR2AHTR1AHTR6DRD2HTR7
SCHEMBL28413707 0.88 HRH3 (0.63) HTR2AHTR1AHTR6DRD2HTR7
SCHEMBL7015692 0.88 HRH3 (0.67) HTR2AHTR1AHTR6DRD2HTR7
SCHEMBL8263255 0.88 HTR2A (0.65) HTR2AHTR1AHTR6DRD2HTR7
SCHEMBL8265592 0.86 MEN1 (0.62) KMT2AHRH3MEN1SMN1; SMN2MAPT
SCHEMBL19778568 0.85 HRH3 (0.67) HTR2AHTR1AHTR6DRD2HTR7
SCHEMBL7011744 0.85 GOT1 (0.70) HTR2AHTR1AHTR6DRD2HTR7
SCHEMBL8264766 0.84 CDK2 (0.61) HTR2AHTR1AHTR6DRD2HTR7
SCHEMBL7006163 0.84 DRD2 (0.73) HTR2AHTR1AHTR6DRD2HTR7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113683552-B Tryptamine salicylic acid compound and preparation and application thereof 兰州大学 2024-03-19 CN disclosed
CN-113683552-A Tryptamine salicylic acid compound and preparation and application thereof 兰州大学 2021-11-23 CN disclosed
CN-107552089-A Application and application process of a kind of quinine squaric amide derivative as asymmetric P S reacting middle catalysts 浙江工业大学 2018-01-09 CN disclosed
EP-1379239-A2 N-(2-ARYLETHYL) BENZYLAMINES AS ANTAGONISTS OF THE 5-HT6 RECEPTOR ELI LILLY AND COMPANY (US) 2004-01-14 EP disclosed
WO-2002078693-A2 N-(2-ARYLETHYL)BENZYLAMINES AS ANTAGONISTS OF THE 5-HT6 RECEPTOR ELI LILLY AND COMPANY (US) 2002-10-10 WO disclosed
US-4372887-A DIURETIC, ANTITHROMBOGENIC, SMOOTH MUSCLE RELAXANTS MEAD JOHNSON & COMPANY (US) 1983-02-08 US disclosed
US-4259238-A ANTIARRHYTHMIA AGENTS MEAD JOHNSON & COMPANY (US) 1981-03-31 US disclosed
US-4196212-A DIURETIC, ANTITHROMBOGENIC, SMOOTH MUSCLE RELAXANT, ANTIINFLAMMATORY MEAD JOHNSON & COMPANY (US) 1980-04-01 US disclosed
US-4091102-A Anti-depressant trans-hexahydropyrido[3,4-b]indoles ENDO LABORATORIES, INC. (US) 1978-05-23 US disclosed
US-4072675-A DIURETICS, ANTICOAGULANTS, INOTROPIC AGENTS, ANTIINFLAMMATORY AGENTS, ANTIARRHYTHMIA AGENTS MEAD JOHNSON & COMPANY (US) 1978-02-07 US disclosed
US-4049714-A DIURETIC, ANTITHROMBOGENIC, ANTIARRYTHMIC, ANTIINFLAMMATORY, MUSCLE RELAXANTS MEAD JOHNSON & COMPANY (US) 1977-09-20 US disclosed