SCHEMBL6600129

SCHEMBL6600129

COc1ccccc1N1CCN(CC/C(=N/O)c2sc3ccccc3c2C)CC1

nearest known ligand 0.66

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 10/20 0.55
HTR1D P28221 2/20 0.55
DRD2 P14416 3/20 0.53
DRD3 P35462 2/20 0.53
DRD4 P21917 1/20 0.52
ADRA1D P25100 2/20 0.50
ADRA1A P35348 2/20 0.50
ADRA1B P35368 2/20 0.50
ALDH1A1 P00352 1/20 0.49
MAPT P10636 1/20 0.49
HTT P42858 1/20 0.49
KMT2A Q03164 1/20 0.49
HTR7 P34969 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6600132 1.00 HTR1A (0.55) HTR1AHTR1DDRD2DRD3DRD4
SCHEMBL7970947 0.91 HTR1A (0.50) HTR1AHTR1DDRD2DRD3DRD4
SCHEMBL7970944 0.91 HTR1A (0.50) HTR1AHTR1DDRD2DRD3DRD4
Hydrochloric Acid SCHEMBL6599492 0.87 HTR1A (0.66) HTR1AHTR1DDRD2DRD3ADRA1D
SCHEMBL6598694 0.81 HTR1A (0.75) HTR1AHTR1DDRD2DRD3DRD4
SCHEMBL6598700 0.81 HTR1A (0.75) HTR1AHTR1DDRD2DRD3DRD4
SCHEMBL8120660 0.81 DRD4 (0.58) HTR1AHTR1DDRD2DRD3DRD4
SCHEMBL6598932 0.79 HTR1A (0.61) HTR1AHTR1DDRD2DRD3DRD4
SCHEMBL6351477 0.79 DRD4 (0.76) HTR1ADRD2DRD3DRD4ADRA1D
SCHEMBL6351475 0.79 DRD4 (0.76) HTR1ADRD2DRD3DRD4ADRA1D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1008594-B1 COMPOUNDS DERIVED FROM THOPHENE AND BENZOTHIOPHENE, AND RELATED UTILISATION AND COMPOSITION VITA LAB (ES) 2004-03-17 EP disclosed
EP-1008594-A1 COMPOUNDS DERIVED FROM THOPHENE AND BENZOTHIOPHENE, AND RELATED UTILISATION AND COMPOSITION VITA-INVEST, S.A. (ES) 2000-06-14 EP disclosed