SCHEMBL6600260

SCHEMBL6600260

NC(=O)c1nc([C@@H](Cc2ccc3ccccc3c2)NC(=O)[C@H](N)Cc2ccc3ccccc3c2)sc1-c1ccccc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSC P53634 1/20 0.45
MME P08473 2/20 0.43
ACE P12821 2/20 0.43
CPA1 P15085 2/20 0.43
ACE2 Q9BYF1 2/20 0.43
OPRD1 P41143 1/20 0.42
PTPN1 P18031 3/20 0.41
PTPN2 P17706 1/20 0.41
PTPN6 P29350 1/20 0.41
CDC25B P30305 1/20 0.41
PTPN11 Q06124 1/20 0.41
FCER2 P06734 1/20 0.40
PTPRB P23467 1/20 0.40
TPH1 P17752 2/20 0.39
DPP4 P27487 1/20 0.39
PRCP P42785 1/20 0.39
NLN Q9BYT8 1/20 0.39
CTSL P07711 1/20 0.38
CTSB P07858 1/20 0.38
CTSS P25774 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27494688 1.00 CTSC (0.45) CTSCMMEACECPA1ACE2
SCHEMBL6602216 0.84 MME (0.42) CTSCMMEACECPA1ACE2
SCHEMBL27493870 0.84 MME (0.42) CTSCMMEACECPA1ACE2
SCHEMBL6599351 0.83 CTSS (0.56) PTPN1PTPRBCTSLCTSBCTSS
SCHEMBL27552033 0.83 CTSS (0.52) PTPN1PTPN2PTPN6CDC25BPTPN11
SCHEMBL6600308 0.83 CTSS (0.52) PTPN1PTPN2PTPN6CDC25BPTPN11
SCHEMBL6600113 0.79 PTPN1 (0.36) MMEACECPA1ACE2PTPN1
SCHEMBL6599339 0.76 CAPN1 (0.44) PTPN1PTPN2PTPN6CDC25BPTPN11
SCHEMBL6600491 0.76 CTSS (0.53) PTPN1PTPN2PTPN6CDC25BPTPN11
SCHEMBL27478624 0.76 CTSS (0.53) PTPN1PTPN2PTPN6CDC25BPTPN11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0805816-B1 COMPOUNDS WITH GROWTH HORMONE RELEASING PROPERTIES NOVO NORDISK AS (DK) 2004-07-28 EP claimed
EP-0805816-B1 COMPOUNDS WITH GROWTH HORMONE RELEASING PROPERTIES NOVO NORDISK AS (DK) 2004-07-28 EP disclosed
US-6350767-B1 GROWTH HORMONE RELEASE STIMULANT NOVO NORDISK A/S (DK) 2002-02-26 US disclosed
US-6013658-A ANIMAL GROWTH REGULATORS NOVO NORDISK A/S (DK) 2000-01-11 US disclosed
EP-0907374-A1 GROWTH HORMONE COMPONENT AND BONE ANTI-RESORPTIVE AGENT IN CYCLIC (COHERENCE) TREATMENT OF OSTEOPOROSIS NOVO NORDISK A/S (DK) 1999-04-14 EP disclosed
CN-1176645-A Compounds with growth hormone releasing properties NOVO NORDISK AS (DK) 1998-03-18 CN disclosed
WO-1997046252-A1 GROWTH HORMONE COMPONENT AND BONE ANTI-RESORPTIVE AGENT IN CYCLIC (COHERENCE) TREATMENT OF OSTEOPOROSIS NOVO NORDISK A/S (DK) 1997-12-11 WO disclosed
WO-1996022997-A1 COMPOUNDS WITH GROWTH HORMONE RELEASING PROPERTIES NOVO NORDISK A/S (DK) 1996-08-01 WO disclosed