SCHEMBL6600262

SCHEMBL6600262

COCc1ccccc1C(=O)Cl

nearest known ligand 0.44

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.44
ALOX15 P16050 1/20 0.44
TSHR P16473 2/20 0.43
HTT P42858 2/20 0.42
TP53 P04637 1/20 0.42
PRMT5 O14744 1/20 0.42
LMNA P02545 2/20 0.41
CTSD P07339 1/20 0.41
HDAC3 O15379 1/20 0.40
HDAC1 Q13547 1/20 0.40
KMT2A Q03164 1/20 0.40
HPGD P15428 1/20 0.39
MRGPRX4 Q96LA9 1/20 0.39
FFAR1 O14842 1/20 0.38
C5AR1 P21730 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11555943 0.85 ALDH1A1 (0.39) ALDH1A1ALOX15TSHRHTTTP53
SCHEMBL16245167 0.84 TSHR (0.46) ALDH1A1ALOX15TSHRHTTTP53
SCHEMBL3145722 0.82 LMNA (0.46) ALDH1A1TSHRHTTTP53PRMT5
SCHEMBL534811 0.82 HTT (0.56) ALDH1A1ALOX15TSHRHTTTP53
SCHEMBL31617745 0.82 HTT (0.56) ALDH1A1ALOX15TSHRHTTTP53
SCHEMBL23292529 0.81 CTSD (0.59) ALDH1A1TSHRPRMT5LMNACTSD
SCHEMBL28343391 0.81 ALDH1A1 (0.52) ALDH1A1ALOX15TSHRHTTTP53
SCHEMBL9259808 0.81 HDAC3 (0.39) ALDH1A1TSHRHTTTP53PRMT5
SCHEMBL9021410 0.81 HDAC3 (0.39) ALDH1A1TSHRHTTTP53PRMT5
SCHEMBL3150175 0.81 ALDH1A1 (0.62) ALDH1A1ALOX15TSHRHTTLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1379525-A2 HETEROPOLYCYCLIC COMPOUNDS AND THEIR USE AS METABOTROPIC GLUTAMATE RECEPTOR ANTAGONISTS NPS PHARMACEUTICALS, INC. (US) 2004-01-14 EP disclosed
WO-2002068417-A3 HETEROPOLYCYCLIC COMPOUNDS AND THEIR USE AS METABOTROPIC GLUTAMATE RECEPTOR ANTAGONISTS SLASSI ABDELMALIK (CA) 2002-11-14 WO disclosed
WO-2002068417-A2 HETEROPOLYCYCLIC COMPOUNDS AND THEIR USE AS METABOTROPIC GLUTAMATE RECEPTOR ANTAGONISTS NPS PHARMACEUTICALS, INC. (US) 2002-09-06 WO disclosed
US-4960943-A ACYLATING REACTION IN THE PRESENCE OF ZEOLITE CATALYSTS BAYER AKTIENGESELLSCHAFT (DE) 1990-10-02 US disclosed
EP-0155792-B1 BENZOATE DERIVATIVES HAVING POSITIVE DIELECTRIC ANISOTROPY AND LIQUID CRYSTAL COMPOSITIONS CONTAINING THEM Chisso Corporation (JP) 1987-06-16 EP disclosed
US-4661283-A Benzoate derivatives having a large positive dielectric anisotropy value and liquid crystal compositions containing same CHISSO CORPORATION (JP) 1987-04-28 US disclosed
EP-0155792-A1 Benzoate derivatives having positive dielectric anisotropy and liquid crystal compositions containing them Chisso Corporation (JP) 1985-09-25 EP disclosed