SCHEMBL6600548

SCHEMBL6600548

CC(C)(C)c1csc(-c2cc3cc(Cn4nc5ccccc5c4-c4nnn[nH]4)ccc3o2)n1

nearest known ligand 0.31

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
TP53 P04637 1/20 0.31
TSHR P16473 1/20 0.31
STAT1 P42224 1/20 0.31
LMNA P02545 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6601175 0.81 TSHR (0.33) TP53TSHRSTAT1LMNA
SCHEMBL6601208 0.80 CCR2 (0.35)
SCHEMBL7476880 0.80 PTGER4 (0.36) TP53TSHRSTAT1
SCHEMBL6600915 0.79 PDE5A (0.34)
SCHEMBL6600027 0.79 PDE5A (0.34)
SCHEMBL6600909 0.78 PDE5A (0.34)
SCHEMBL6597519 0.77
SCHEMBL6597036 0.76 CNR1 (0.33)
SCHEMBL6598376 0.76 PTGER4 (0.39)
SCHEMBL8659965 0.74 MEN1 (0.40) TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1170009-B1 Thiazolybenzofuran derivatives and their use as SRS-A and leukotiene antagonists FUJISAWA PHARMACEUTICAL CO (JP) 2004-04-07 EP disclosed
EP-1170009-A2 Thiazolybenzofuran derivatives and their use as SRS-A and leukotiene antagonists FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2002-01-09 EP disclosed
US-5994378-A ANTIALLERGENS; ANTIINFLAMMATORY AGENTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1999-11-30 US disclosed