SCHEMBL6600673

SCHEMBL6600673

CC(C)(C)OC(=O)N1CCC(c2cn(-c3ccc(F)cc3)c3ccccc23)CC1

nearest known ligand 0.52

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 2/20 0.52
TP53 P04637 2/20 0.50
GPR119 Q8TDV5 3/20 0.49
ALDH1A1 P00352 2/20 0.49
LMNA P02545 2/20 0.49
MEN1 O00255 1/20 0.48
KMT2A Q03164 1/20 0.48
POLB P06746 1/20 0.48
CYP3A4 P08684 1/20 0.46
CYP2D6 P10635 1/20 0.46
CYP2C9 P11712 1/20 0.46
CYP2C19 P33261 1/20 0.46
SCN9A Q15858 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14406151 0.90 GPR119 (0.47) GPR119ALDH1A1LMNASCN9A
SCHEMBL6598945 0.86 DRD2 (0.47) KCNH2ALDH1A1LMNAPOLBCYP3A4
SCHEMBL19972594 0.86 GPR119 (0.50) TP53GPR119ALDH1A1LMNAPOLB
SCHEMBL6966415 0.84 GPR119 (0.47) KCNH2GPR119
SCHEMBL6600804 0.84 HTR1B (0.60)
SCHEMBL6601681 0.82 DRD2 (0.70) GPR119POLB
SCHEMBL6600206 0.82 DRD2 (0.71) GPR119
SCHEMBL558066 0.82 SCN9A (0.61) TP53GPR119MEN1KMT2ASCN9A
SCHEMBL6603834 0.81 DRD2 (0.71) GPR119POLB
SCHEMBL27322905 0.81 SCN9A (0.50) GPR119MEN1KMT2ASCN9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1478643-A1 5-HETEROARYL SUBSTITUTED INDOLES H. Lundbeck A/S (DK) 2004-11-24 EP disclosed
WO-2003070723-A1 5-HETEROARYL SUBSTITUTED INDOLES H. LUNDBECK A/S (DK) 2003-08-28 WO disclosed