SCHEMBL6600917

SCHEMBL6600917

CC(C)(C)OC(=O)NC1(C(=O)NC2C(O)CCCCN2C(=O)OCc2ccccc2)CCCCC1

nearest known ligand 0.45

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CTSS P25774 6/20 0.45
CTSL P07711 5/20 0.45
CTSB P07858 4/20 0.45
CTSK P43235 5/20 0.45
FKBP1A P62942 5/20 0.43
PDE4B Q07343 1/20 0.41
TMEM97 Q5BJF2 2/20 0.40
SIGMAR1 Q99720 2/20 0.40
KMT2A Q03164 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
PDK1 Q15118 1/20 0.39
PDK2 Q15119 1/20 0.39
PDK3 Q15120 1/20 0.39
PDK4 Q16654 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6604451 0.83 CTSS (0.44) CTSSCTSLCTSBCTSKPDE4B
SCHEMBL6600419 0.82 CTSK (0.44) CTSSCTSLCTSBCTSKFKBP1A
SCHEMBL30804803 0.78 KLK7 (0.48) CTSLCTSBCTSKFKBP1AKMT2A
SCHEMBL27512771 0.78 CTSK (0.57) CTSSCTSLCTSBCTSK
SCHEMBL27978282 0.77 FKBP1A (0.52) CTSSCTSLCTSBCTSKFKBP1A
SCHEMBL1449131 0.77 CTSL (0.47) CTSSCTSLCTSBPDE4BKMT2A
SCHEMBL29080198 0.76 CTSL (0.46) CTSSCTSLCTSBCTSKPDE4B
SCHEMBL30860130 0.75 CTSL (0.46) CTSSCTSLCTSBCTSKPDE4B
SCHEMBL30793744 0.75 CTSL (0.45) CTSSCTSLCTSBCTSKPDE4B
SCHEMBL550418 0.75 CTSL (0.56) CTSSCTSLCTSBCTSKKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1392657-A4 PROTEASE INHIBITORS SMITHKLINE BEECHAM CORP (US) 2004-03-10 EP disclosed
EP-1392657-A2 PROTEASE INHIBITORS SmithKline Beecham Corporation (US) 2004-03-03 EP disclosed
WO-2003053331-A2 PROTEASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2003-07-03 WO disclosed