SCHEMBL6603385

SCHEMBL6603385

CCOC(=O)c1ccc(NC(=O)OCc2c[nH]c(-c3cc4nc(C(=O)OCC)c(OCC)nc4cc3[N+](=O)[O-])n2)c(F)c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.40
ALDH1A1 P00352 7/20 0.39
KDM4E B2RXH2 1/20 0.39
POLB P06746 1/20 0.39
MAPT P10636 7/20 0.38
RAB9A P51151 4/20 0.38
NPC1 O15118 3/20 0.38
PKM P14618 1/20 0.38
CRHBP P24387 1/20 0.38
CRHR2 Q13324 1/20 0.38
LMNA P02545 1/20 0.37
PTGER4 P35408 1/20 0.36
SMN1; SMN2 Q16637 4/20 0.34
MEN1 O00255 3/20 0.34
TP53 P04637 2/20 0.34
HPGD P15428 2/20 0.34
NPSR1 Q6W5P4 1/20 0.33
THRB P10828 1/20 0.33
GRIA1 P42261 1/20 0.33
GRIA2 P42262 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6602557 0.94 KMT2A (0.38) KMT2AALDH1A1KDM4EPOLBMAPT
SCHEMBL6602436 0.90 ALDH1A1 (0.41) KMT2AALDH1A1KDM4EPOLBMAPT
SCHEMBL6601960 0.87 KMT2A (0.41) KMT2AALDH1A1KDM4EPOLBMAPT
SCHEMBL6603788 0.85 ALDH1A1 (0.38) KMT2AALDH1A1POLBMAPTLMNA
SCHEMBL6603403 0.81 MAPT (0.32) KMT2AALDH1A1KDM4EPOLBMAPT
SCHEMBL6603534 0.81 ALDH1A1 (0.36) KMT2AALDH1A1KDM4EPOLBMAPT
SCHEMBL6604561 0.81 ALDH1A1 (0.39) KMT2AALDH1A1KDM4EPOLBMAPT
SCHEMBL6605470 0.78 ALDH1A1 (0.34) KMT2AALDH1A1KDM4EPOLBMAPT
SCHEMBL6382753 0.78 NAMPT (0.43) KMT2AKDM4EPOLBMAPTRAB9A
SCHEMBL6631139 0.77 ALDH1A1 (0.40) KMT2AALDH1A1KDM4EPOLBMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1020453-B1 6,7-ASYMMETRICALLY DISUBSTITUTED QUINOXALINECARBOXYLIC ACID DERIVATIVES, ADDITION SALTS THEREOF, AND PROCESSES FOR THE PREPARATION OF BOTH KYORIN SEIYAKU KK (JP) 2004-05-19 EP disclosed
US-6348461-B1 CENTRAL NERVOUS SYSTEM ANTAGONIST WITH HETEROCYCLIC SUBSTITUENTS KYORIN PHARMACEUTICAL CO., LTD. (JP) 2002-02-19 US disclosed
EP-1020453-A1 6,7-ASYMMETRICALLY DISUBSTITUTED QUINOXALINECARBOXYLIC ACID DERI VATIVES, ADDITION SALTS THEREOF, AND PROCESSES FOR THE PREPARATION OF BOTH KYORIN PHARMACEUTICAL CO., LTD. (JP) 2000-07-19 EP disclosed