SCHEMBL6607104

SCHEMBL6607104

CCCCCCc1cc(C(=O)O)nc2c(OCc3ccccc3)cccc12

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGER1 P34995 4/20 0.45
PPARA Q07869 3/20 0.45
MRGPRX4 Q96LA9 2/20 0.44
FOLH1 Q04609 1/20 0.44
BCHE P06276 2/20 0.44
PPARG P37231 2/20 0.43
PTGER4 P35408 2/20 0.43
PTGER3 P43115 2/20 0.43
PTGER2 P43116 2/20 0.43
HDAC3 O15379 2/20 0.42
HDAC4 P56524 2/20 0.42
HDAC1 Q13547 2/20 0.42
HDAC7 Q8WUI4 2/20 0.42
HDAC2 Q92769 2/20 0.42
HDAC10 Q969S8 2/20 0.42
HDAC11 Q96DB2 2/20 0.42
HDAC8 Q9BY41 2/20 0.42
HDAC6 Q9UBN7 2/20 0.42
HDAC9 Q9UKV0 2/20 0.42
HDAC5 Q9UQL6 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6079710 0.92 MTNR1A (0.43) PTGER1PPARABCHEHDAC3HDAC4
SCHEMBL6599193 0.90 HDAC3 (0.45) PTGER1MRGPRX4FOLH1PTGER4PTGER3
SCHEMBL6590566 0.87 MRGPRX4 (0.46) PTGER1MRGPRX4FOLH1PTGER4PTGER3
SCHEMBL6079754 0.84 HDAC3 (0.44) PTGER1MRGPRX4FOLH1PTGER4PTGER3
SCHEMBL6593195 0.82 MTNR1B (0.56) PTGER1MRGPRX4PTGER4PTGER3PTGER2
SCHEMBL6597561 0.81 MTNR1A (0.43) PTGER1BCHEHDAC3HDAC4HDAC1
SCHEMBL6080597 0.81 ADORA3 (0.41) PTGER1MRGPRX4FOLH1PTGER4PTGER3
SCHEMBL6079714 0.80 ADORA1 (0.43) PTGER1PPARAMRGPRX4FOLH1BCHE
SCHEMBL6596257 0.80 CTSL (0.43) PTGER1MRGPRX4FOLH1HDAC3HDAC4
SCHEMBL6080497 0.79 MRGPRX4 (0.51) PTGER1MRGPRX4FOLH1HDAC3HDAC4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1451159-A1 COMPOSITIONS DERIVED FROM QUINOLINE AND QUINOXALINE, PREPARATION AND USE THEREOF NEURO3D (FR) 2004-09-01 EP disclosed
WO-2003010146-A1 COMPOSITIONS DERIVED FROM QUINOLINE AND QUINOXALINE, PREPARATION AND USE THEREOF NEURO3D (FR) 2003-02-06 WO disclosed