SCHEMBL6607169

SCHEMBL6607169

O=C(O)CC(NC(=O)c1ccc(C(F)(F)F)cc1)C(=O)CF

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA2 P00918 2/20 0.47
CA1 P00915 1/20 0.47
PTPN1 P18031 1/20 0.44
CASP3 P42574 9/20 0.43
NPC1 O15118 1/20 0.42
RAB9A P51151 1/20 0.42
CES2 O00748 1/20 0.42
CES1 P23141 1/20 0.42
TMPRSS15 P98073 1/20 0.42
LMNA P02545 1/20 0.41
SRD5A2 P31213 1/20 0.41
PIN1 Q13526 1/20 0.41
CASP7 P55210 1/20 0.41
CASP9 P55211 1/20 0.41
CASP6 P55212 1/20 0.41
CASP8 Q14790 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2C9 P11712 1/20 0.41
TSHR P16473 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6609413 0.85 NPSR1 (0.58) CES2LMNAPIN1
SCHEMBL6607173 0.85 CASP3 (0.52) CA2CA1CASP3NPC1
SCHEMBL6606162 0.85 CASP3 (0.52) CA2CA1CASP3CASP7CASP9
SCHEMBL6607828 0.84 CASP3 (0.53) CA2CA1CASP3LMNACASP7
SCHEMBL6610883 0.84 HPGDS (0.53) CA2CA1CASP3NPC1RAB9A
SCHEMBL6607165 0.84 CASP3 (0.52) CA2CA1CASP3LMNA
SCHEMBL6606242 0.81 MEN1 (0.49) CA2CA1CASP3
SCHEMBL6606122 0.81 TAS1R3 (0.51) CA2CA1CASP3CYP3A4
SCHEMBL6606153 0.80 CA2 (0.44) CA2CA1CASP3CASP7CASP9
SCHEMBL6609614 0.78 GRN (0.56) CA2CA1CASP3CYP1A2CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1163208-B1 CASPASE INHIBITORS AND USES THEREOF VERTEX PHARMA (US) 2004-05-12 EP disclosed