SCHEMBL6607734

SCHEMBL6607734

CC1=C(C#N)C(c2cccc(-c3ccc(Cl)cc3)c2)NC(=O)N1C(=O)O

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ELANE P08246 1/20 0.37
CYP2C9 P11712 1/20 0.37
GRIA2 P42262 3/20 0.36
GRIA4 P48058 3/20 0.36
MAPT P10636 2/20 0.36
HTT P42858 2/20 0.35
ALDH1A1 P00352 3/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
HTR2C P28335 1/20 0.34
HSD17B3 P37058 2/20 0.34
SHMT1 P34896 1/20 0.34
SHMT2 P34897 1/20 0.34
LMNA P02545 2/20 0.33
CNR1 P21554 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
KDM4E B2RXH2 1/20 0.33
GAA P10253 1/20 0.33
RAD51 Q06609 1/20 0.33
CHEK1 O14757 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6137118 0.88 HTT (0.43) ELANECYP2C9MAPTHTTALDH1A1
SCHEMBL6608315 0.88 ELANE (0.37) ELANECYP2C9MAPTALDH1A1MEN1
SCHEMBL6610688 0.84 DRD2 (0.39) ELANECYP2C9HTTMEN1KMT2A
SCHEMBL6608080 0.84 ALDH1A1 (0.40) ELANECYP2C9MAPTHTTALDH1A1
SCHEMBL6609236 0.82 ELANE (0.45) ELANECYP2C9TDP1
SCHEMBL6137166 0.82 KMT2A (0.45) ELANECYP2C9HTTALDH1A1MEN1
SCHEMBL6608143 0.82 ALOX5 (0.39) ELANECYP2C9MAPTMEN1KMT2A
SCHEMBL6608283 0.81 ELANE (0.40) ELANECYP2C9MAPTALDH1A1MEN1
SCHEMBL6137365 0.81 ELANE (0.40) ELANECYP2C9MAPTHTTALDH1A1
SCHEMBL6608090 0.81 MAPK1 (0.44) ELANECYP2C9MAPTHTTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1373223-A4 CYANO-SUBSTITUTED DIHYDROPYRIMIDINE COMPOUNDS AND THEIR USE TO TREAT DISEASES BRISTOL MYERS SQUIBB CO (US) 2004-09-29 EP disclosed
EP-1373223-A1 CYANO-SUBSTITUTED DIHYDROPYRIMIDINE COMPOUNDS AND THEIR USE TO TREAT DISEASES Bristol-Myers Squibb Company (US) 2004-01-02 EP disclosed
WO-2002079169-A1 CYANO-SUBSTITUTED DIHYDROPYRIMIDINE COMPOUNDS AND THEIR USE TO TREAT DISEASES BRISTOL-MYERS SQUIBB COMPANY (US) 2002-10-10 WO disclosed