SCHEMBL6608117

SCHEMBL6608117

Nc1cc(Cl)c(NCC2CC2)cc1NC(=O)O

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGER4 P35408 3/20 0.47
KDM4C Q9H3R0 3/20 0.41
LIPC P11150 1/20 0.39
LIPG Q9Y5X9 1/20 0.39
PIK3C3 Q8NEB9 1/20 0.36
VCP P55072 2/20 0.36
HDAC3 O15379 1/20 0.36
HDAC1 Q13547 1/20 0.36
HDAC2 Q92769 1/20 0.36
KDM4E B2RXH2 1/20 0.35
ASPH Q12797 1/20 0.35
RIOX2 Q8IUF8 1/20 0.35
KDM8 Q8N371 1/20 0.35
CNR2 P34972 1/20 0.35
CRHR1 P34998 2/20 0.35
SCN5A Q14524 3/20 0.35
CYP3A4 P08684 2/20 0.35
SCN9A Q15858 2/20 0.35
NPC1 O15118 1/20 0.35
RAB9A P51151 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6165854 0.81 PTGER4 (0.44) PTGER4HDAC3HDAC1HDAC2
SCHEMBL6607350 0.80 LIPC (0.47) PTGER4KDM4CLIPCLIPGPIK3C3
SCHEMBL6641223 0.79 L3MBTL1 (0.44) PTGER4KDM4ENPC1RAB9A
SCHEMBL27615952 0.76 MEN1 (0.43) KDM4CHDAC1KDM4ENPC1RAB9A
SCHEMBL1726529 0.71 PRKCI (0.41) HDAC1KDM4ENPC1RAB9APOLB
SCHEMBL27597105 0.71 CD44 (0.52) HDAC3HDAC1HDAC2KDM4ECYP3A4
SCHEMBL3930758 0.70 PTGER4 (0.51) PTGER4KDM4CLIPCLIPGKDM4E
SCHEMBL15774700 0.70 PTGER4 (0.67) PTGER4KDM4CLIPCLIPGKDM4E
SCHEMBL30102420 0.69 PTGER4 (0.41) PTGER4KDM4CKDM4EASPHRIOX2
SCHEMBL27270334 0.69 PTGER4 (0.55) PTGER4LIPCLIPGVCPCNR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1379511-A1 DIHYDRO-BENZO (b) (1, 4) DIAZEPIN-2-ONE DERIVATIVES AS MGLUR2 ANTAGONISTS II F. HOFFMANN-LA ROCHE AG (CH) 2004-01-14 EP disclosed
WO-2002083652-A1 DIHYDRO-BENZO [b] [1, 4] DIAZEPIN-2-ONE DERIVATIVES AS MGLUR2 ANTAGONISTS II F. HOFFMANN-LA ROCHE AG (CH) 2002-10-24 WO disclosed