SCHEMBL6608915

SCHEMBL6608915

CCCN(Cc1ccc(-c2ccccc2C#N)cc1)c1nc2ccccc2cc1C(=O)OCC

nearest known ligand 0.42

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
AGTR1 P30556 12/20 0.42
AGTR2 P50052 12/20 0.42
KDM4E B2RXH2 6/20 0.41
ALDH1A1 P00352 6/20 0.41
TDP1 Q9NUW8 5/20 0.41
L3MBTL1 Q9Y468 5/20 0.41
LMNA P02545 3/20 0.41
HPGD P15428 3/20 0.41
NPSR1 Q6W5P4 1/20 0.41
HSD17B10 Q99714 1/20 0.40
PPARG P37231 1/20 0.40
HTT P42858 1/20 0.40
GPR55 Q9Y2T6 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6611120 0.86 AGTR1 (0.55) AGTR1AGTR2ALDH1A1
SCHEMBL6606838 0.83 AGTR1 (0.53) AGTR1AGTR2KDM4EALDH1A1TDP1
SCHEMBL8944453 0.83 AGTR1 (0.46) AGTR1AGTR2
SCHEMBL6604855 0.81 AGTR1 (0.43) AGTR1AGTR2
SCHEMBL6608525 0.81 AGTR1 (0.44) AGTR1AGTR2
SCHEMBL8552171 0.79 MAP2K1 (0.40) AGTR1AGTR2KDM4EALDH1A1TDP1
SCHEMBL6606990 0.79 AGTR1 (0.57) AGTR1AGTR2
SCHEMBL9542915 0.78 AGT (0.46) AGTR1AGTR2
SCHEMBL9409377 0.76 AGTR1 (0.40) AGTR1AGTR2KDM4EALDH1A1HSD17B10
SCHEMBL9424056 0.76 AGTR1 (0.67) AGTR1AGTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0829479-B1 Heterocyclic compounds and their use as angiotensin II antagonists TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2004-04-14 EP disclosed
EP-0588299-B1 1,2,4-Oxadiazolyl- or 1,2,4-thiadiazolyl-biphenyl derivatives as angiotensin II antagonists TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1998-07-01 EP disclosed
EP-0829479-A1 Heterocyclic compounds and their use as angiotensin II antagonists TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-03-18 EP disclosed
US-5500427-A ANGIOTENSIN II ANTAGONISTS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-03-19 US disclosed
EP-0588299-A2 1,2,4-Oxadiazolyl- or 1,2,4-thiadiazolyl-biphenyl derivatives as angiotensin II antagonists TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1994-03-23 EP disclosed