SCHEMBL9409377

SCHEMBL9409377

CCCN(Cc1ccc(-c2ccccc2C#N)cc1)c1[nH]nc(C)c1C(=O)OCC

nearest known ligand 0.40

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
AGTR1 P30556 18/20 0.40
AGTR2 P50052 18/20 0.40
PDE4D Q08499 1/20 0.37
KDM4E B2RXH2 1/20 0.37
ALDH1A1 P00352 1/20 0.37
HSD17B10 Q99714 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6606838 0.77 AGTR1 (0.53) AGTR1AGTR2KDM4EALDH1A1HSD17B10
SCHEMBL6611120 0.76 AGTR1 (0.55) AGTR1AGTR2ALDH1A1
SCHEMBL6608915 0.76 AGTR1 (0.42) AGTR1AGTR2KDM4EALDH1A1HSD17B10
SCHEMBL8552171 0.76 MAP2K1 (0.40) AGTR1AGTR2KDM4EALDH1A1HSD17B10
SCHEMBL9409382 0.75 KDM4E (0.39) KDM4EALDH1A1HSD17B10
SCHEMBL6606990 0.73 AGTR1 (0.57) AGTR1AGTR2
SCHEMBL9424056 0.71 AGTR1 (0.67) AGTR1AGTR2
SCHEMBL7810041 0.69
SCHEMBL2730 0.68 LTB4R2 (0.53) AGTR1
SCHEMBL8553595 0.67 LTB4R2 (0.45) AGTR1AGTR2KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0588299-A2 1,2,4-Oxadiazolyl- or 1,2,4-thiadiazolyl-biphenyl derivatives as angiotensin II antagonists TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1994-03-23 EP disclosed