SCHEMBL6609038

SCHEMBL6609038

CN(C)c1cc(NC(=O)O)c(NC(=O)CC(=O)c2cccc(-c3cc(COC4CCCCO4)nn3C)c2)cc1Cl

nearest known ligand 0.34

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
SLC16A3 O15427 11/20 0.34
SLC16A1 P53985 11/20 0.34
CREBBP Q92793 2/20 0.34
EP300 Q09472 1/20 0.34
MCTS1 Q9ULC4 5/20 0.33
RORC P51449 2/20 0.32
FAAH O00519 1/20 0.32
EIF4EBP1 Q13541 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6163574 0.93 SLC16A3 (0.33) SLC16A3SLC16A1CREBBPEP300MCTS1
SCHEMBL6606146 0.84 CREBBP (0.33) CREBBPEP300
SCHEMBL6609371 0.82 CREBBP (0.38) SLC16A3SLC16A1CREBBPEP300MCTS1
SCHEMBL6609350 0.80 HSD11B1 (0.36) CREBBPEP300RORC
SCHEMBL6607850 0.80 CREBBP (0.39) CREBBPEP300
SCHEMBL6163707 0.80 USP30 (0.36)
SCHEMBL6608414 0.78 NTRK1 (0.33) CREBBPEP300RORC
SCHEMBL6164800 0.78 USP30 (0.37) SLC16A3SLC16A1CREBBPEP300MCTS1
SCHEMBL6164138 0.77 NPC1 (0.32) CREBBPEP300
SCHEMBL6165370 0.77 SLC6A9 (0.33) CREBBPEP300

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1379511-A1 DIHYDRO-BENZO (b) (1, 4) DIAZEPIN-2-ONE DERIVATIVES AS MGLUR2 ANTAGONISTS II F. HOFFMANN-LA ROCHE AG (CH) 2004-01-14 EP disclosed
WO-2002083652-A1 DIHYDRO-BENZO [b] [1, 4] DIAZEPIN-2-ONE DERIVATIVES AS MGLUR2 ANTAGONISTS II F. HOFFMANN-LA ROCHE AG (CH) 2002-10-24 WO disclosed