SCHEMBL6609478

SCHEMBL6609478

O=C(Nc1ccc(N(Cc2ccccc2)c2ccccc2)cc1)OC1CC(=O)N(C2Cc3ccccc3C2)C1

nearest known ligand 0.48

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
BCHE P06276 9/20 0.48
ACHE P22303 3/20 0.47
MAOB P27338 2/20 0.42
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38
LMNA P02545 2/20 0.38
HTT P42858 2/20 0.38
ALDH1A1 P00352 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
NR3C2 P08235 1/20 0.37
NAMPT P43490 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6616272 0.90 BCHE (0.47) BCHEACHEMAOBNPC1RAB9A
SCHEMBL6610332 0.89 BCHE (0.49) BCHEACHEMAOBNPC1RAB9A
SCHEMBL6608839 0.86 BCHE (0.50) BCHEACHENPC1RAB9ALMNA
SCHEMBL6610605 0.84 ACHE (0.49) BCHEACHENPC1RAB9AALDH1A1
SCHEMBL5842367 0.83 ALDH1A1 (0.54) NPC1RAB9ALMNAHTTALDH1A1
SCHEMBL6609227 0.83 BCHE (0.55) BCHEACHEMAOBNPC1RAB9A
SCHEMBL6611305 0.83 BCHE (0.59) BCHEACHEMAOBNPC1RAB9A
SCHEMBL6615517 0.79 ALOX15 (0.47) BCHEACHEMAOBLMNAHTT
SCHEMBL6611162 0.79 BCHE (0.39) BCHEMAOBLMNAHTTALDH1A1
SCHEMBL6613814 0.77 MAPT (0.38) BCHEMAOBLMNAALDH1A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1463724-A1 PYRROLIDONE CARBOXAMIDES Actelion Pharmaceuticals Ltd. (CH) 2004-10-06 EP disclosed
WO-2003059905-A1 PYRROLIDONE CARBOXAMIDES ACTELION PHARMACEUTICALS LTD (CH) 2003-07-24 WO disclosed