SCHEMBL6608839

SCHEMBL6608839

CN(c1ccccc1)c1ccc(NC(=O)OC2CC(=O)N(C3Cc4ccccc4C3)C2)cc1

nearest known ligand 0.50

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
BCHE P06276 6/20 0.50
ACHE P22303 4/20 0.50
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
NPY5R Q15761 1/20 0.39
LTA4H P09960 1/20 0.39
CHRNA7 P36544 2/20 0.38
ALDH1A1 P00352 2/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
LMNA P02545 1/20 0.38
MC4R P32245 1/20 0.38
KDM4E B2RXH2 1/20 0.38
MEN1 O00255 1/20 0.38
MAPT P10636 1/20 0.38
THRB P10828 1/20 0.38
GFER P55789 1/20 0.38
KMT2A Q03164 1/20 0.38
TDP1 Q9NUW8 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6610605 0.92 ACHE (0.49) BCHEACHENPC1RAB9ANPY5R
SCHEMBL6616272 0.89 BCHE (0.47) BCHEACHENPC1RAB9AALDH1A1
SCHEMBL6613611 0.87 ACHE (0.42) BCHEACHENPC1RAB9AALDH1A1
SCHEMBL6610332 0.86 BCHE (0.49) BCHEACHENPC1RAB9ACHRNA7
SCHEMBL6609478 0.86 BCHE (0.48) BCHEACHENPC1RAB9AALDH1A1
SCHEMBL6609227 0.86 BCHE (0.55) BCHEACHENPC1RAB9ACHRNA7
SCHEMBL6611305 0.86 BCHE (0.59) BCHEACHENPC1RAB9ACHRNA7
SCHEMBL5842752 0.82 ALDH1A1 (0.58) ALDH1A1SMN1; SMN2LMNAKDM4EMEN1
SCHEMBL6609671 0.79 BCHE (0.47) BCHEACHENPC1RAB9AALDH1A1
SCHEMBL6611149 0.79 MGLL (0.57) BCHEACHENPC1RAB9AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1463724-A1 PYRROLIDONE CARBOXAMIDES Actelion Pharmaceuticals Ltd. (CH) 2004-10-06 EP disclosed
WO-2003059905-A1 PYRROLIDONE CARBOXAMIDES ACTELION PHARMACEUTICALS LTD (CH) 2003-07-24 WO disclosed