SCHEMBL6609843

SCHEMBL6609843

O=C1C(Cc2ccccc2)NC(=O)C2(CCN(c3ccccc3)CC2)N1CCc1c[nH]c2ccccc12

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CXCR3 P49682 1/20 0.49
DRD2 P14416 2/20 0.47
DRD4 P21917 2/20 0.47
DRD3 P35462 2/20 0.47
HTR1A P08908 1/20 0.47
HTR2A P28223 1/20 0.47
SLC6A4 P31645 1/20 0.47
HRH1 P35367 1/20 0.47
HTR2B P41595 1/20 0.47
KMT2A Q03164 3/20 0.46
MEN1 O00255 2/20 0.43
TP53 P04637 1/20 0.42
GLA P06280 1/20 0.42
CYP3A4 P08684 1/20 0.42
MAPT P10636 1/20 0.42
THRB P10828 1/20 0.42
IDO1 P14902 1/20 0.42
RIPK1 Q13546 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
HSD17B10 Q99714 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6617457 0.95 DRD2 (0.50) CXCR3DRD2DRD4DRD3HTR1A
SCHEMBL6613040 0.93 KMT2A (0.50) CXCR3DRD2DRD4DRD3HTR1A
SCHEMBL6617413 0.91 CXCR3 (0.53) CXCR3DRD2DRD4DRD3HTR1A
SCHEMBL6612281 0.91 DRD2 (0.45) CXCR3DRD2DRD4DRD3HTR1A
SCHEMBL6614723 0.89 CXCR3 (0.54) CXCR3DRD2DRD4DRD3HTR1A
SCHEMBL6612079 0.88 CCR5 (0.53) CXCR3DRD2DRD4DRD3HTR1A
SCHEMBL6610512 0.88 CCR5 (0.52) CYP3A4CCR5CXCR4
SCHEMBL6614855 0.87 KMT2A (0.57) CXCR3DRD2DRD4DRD3KMT2A
SCHEMBL6644502 0.87 CCR5 (0.57) CXCR3DRD2DRD4DRD3HTR1A
SCHEMBL6612813 0.86 CXCR3 (0.52) CXCR3DRD2DRD4DRD3HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1236726-B1 TRIAZASPIRO 5.5]UNDECANE DERIVATIVES AND DRUGS CONTAINING THE SAME AS THE ACTIVE INGREDIENT ONO PHARMACEUTICAL CO (JP) 2004-12-01 EP disclosed
EP-1236726-A1 TRIAZASPIRO 5.5]UNDECANE DERIVATIVES AND DRUGS CONTAINING THE SAME AS THE ACTIVE INGREDIENT ONO PHARMACEUTICAL CO., LTD. (JP) 2002-09-04 EP disclosed