SCHEMBL6612281

SCHEMBL6612281

O=C1C(COCc2ccccc2)NC(=O)C2(CCN(c3ccccc3)CC2)N1CCc1c[nH]c2ccccc12

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 2/20 0.45
DRD4 P21917 2/20 0.45
DRD3 P35462 2/20 0.45
HTR1A P08908 1/20 0.45
HTR2A P28223 1/20 0.45
SLC6A4 P31645 1/20 0.45
HRH1 P35367 1/20 0.45
HTR2B P41595 1/20 0.45
HTR1D P28221 3/20 0.41
HTR1B P28222 3/20 0.41
HTR7 P34969 1/20 0.40
SSTR4 P31391 1/20 0.40
SSTR5 P35346 1/20 0.40
CXCR3 P49682 1/20 0.40
CCR5 P51681 7/20 0.40
KMT2A Q03164 2/20 0.39
KDM4E B2RXH2 1/20 0.39
MEN1 O00255 1/20 0.39
ALDH1A1 P00352 1/20 0.39
LMNA P02545 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6611736 0.91 CCR5 (0.44) DRD2DRD4DRD3HTR1AHTR2A
SCHEMBL6609843 0.91 CXCR3 (0.49) DRD2DRD4DRD3HTR1AHTR2A
SCHEMBL6613849 0.90 CCR5 (0.47) DRD2DRD4DRD3HTR1AHTR2A
SCHEMBL6616667 0.90 CXCR3 (0.51) CXCR3CCR5
SCHEMBL6614296 0.89 CCR5 (0.52) DRD2DRD4DRD3HTR1AHTR2A
SCHEMBL6617457 0.89 DRD2 (0.50) DRD2DRD4DRD3HTR1AHTR2A
SCHEMBL6616691 0.88 CCR5 (0.51) DRD2DRD4DRD3HTR1AHTR2A
SCHEMBL6617828 0.88 CCR5 (0.55) DRD2DRD4DRD3HTR1AHTR2A
SCHEMBL6611728 0.87 CCR5 (0.47) CXCR3CCR5CXCR4
SCHEMBL6613040 0.87 KMT2A (0.50) DRD2DRD4DRD3HTR1AHTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1236726-B1 TRIAZASPIRO 5.5]UNDECANE DERIVATIVES AND DRUGS CONTAINING THE SAME AS THE ACTIVE INGREDIENT ONO PHARMACEUTICAL CO (JP) 2004-12-01 EP disclosed
EP-1236726-A1 TRIAZASPIRO 5.5]UNDECANE DERIVATIVES AND DRUGS CONTAINING THE SAME AS THE ACTIVE INGREDIENT ONO PHARMACEUTICAL CO., LTD. (JP) 2002-09-04 EP disclosed