SCHEMBL6610

SCHEMBL6610

Cc1noc(-c2ccc(-c3ccc(CCC(=O)O)cc3)cc2)c1N(C)CCCc1cccc(Cl)c1

nearest known ligand 0.43

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
FFAR1 O14842 8/20 0.43
FFAR4 Q5NUL3 2/20 0.43
DGAT1 O75907 1/20 0.41
AOC3 Q16853 1/20 0.39
NR1H4 Q96RI1 1/20 0.38
PPARD Q03181 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
RXRA P19793 1/20 0.38
RXRB P28702 1/20 0.38
RXRG P48443 1/20 0.38
TP53 P04637 2/20 0.38
MDM2 Q00987 2/20 0.38
PLAAT3 P53816 1/20 0.37
PLAAT5 Q96KN8 1/20 0.37
PLAAT2 Q9NWW9 1/20 0.37
PLAAT4 Q9UL19 1/20 0.37
PPARG P37231 1/20 0.37
ALDH1A1 P00352 1/20 0.37
KMT2A Q03164 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6857 0.92 LPAR1 (0.42) FFAR1FFAR4AOC3NR1H4PPARD
SCHEMBL6934 0.87 FFAR4 (0.46) FFAR1FFAR4PPARDRXRARXRB
SCHEMBL7216 0.85 MAOB (0.41) AOC3SMN1; SMN2ALDH1A1KMT2A
SCHEMBL6150 0.85 BRD4 (0.36) FFAR4AOC3TP53ALDH1A1
SCHEMBL1630 0.84 ABCC3 (0.42) AOC3NR1H4TP53KMT2A
SCHEMBL7466 0.81 LPAR1 (0.47) PPARDPPARG
SCHEMBL1568 0.81 KCNA3 (0.39) AOC3ALDH1A1
SCHEMBL6765 0.79 BRD4 (0.33) AOC3SMN1; SMN2ALDH1A1KMT2A
SCHEMBL6811 0.79 HDAC1 (0.42) FFAR4PPARDRXRARXRBRXRG
SCHEMBL6543 0.77 HDAC1 (0.40) FFAR1FFAR4ALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2483252-A2 COMPOUNDS AS LYSOPHOSPHATIDIC ACID RECEPTOR ANTAGONISTS Amira Pharmaceuticals, Inc. (US) 2012-08-08 EP claimed
WO-2011041694-A2 COMPOUNDS AS LYSOPHOSPHATIDIC ACID RECEPTOR ANTAGONISTS AMIRA PHARMACEUTICALS, INC. (US) 2011-04-07 WO claimed
EP-2483252-A2 COMPOUNDS AS LYSOPHOSPHATIDIC ACID RECEPTOR ANTAGONISTS Amira Pharmaceuticals, Inc. (US) 2012-08-08 EP disclosed
WO-2011041694-A2 COMPOUNDS AS LYSOPHOSPHATIDIC ACID RECEPTOR ANTAGONISTS AMIRA PHARMACEUTICALS, INC. (US) 2011-04-07 WO disclosed