SCHEMBL6610889

SCHEMBL6610889

O=C(Cc1cscc1NS(=O)(=O)c1c(Cl)cc(Cl)cc1Cl)N1CCSCC1

nearest known ligand 0.52

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 4/20 0.52
SLC40A1 Q9NP59 1/20 0.35
CNR1 P21554 6/20 0.35
ITGAV P06756 1/20 0.35
MAPK1 P28482 1/20 0.34
CCKBR P32239 1/20 0.34
ACLY P53396 1/20 0.33
HSD17B1 P14061 1/20 0.33
HSD17B2 P37059 1/20 0.33
RORC P51449 1/20 0.33
ALDH1A1 P00352 1/20 0.32
HPGD P15428 1/20 0.32
HSD17B10 Q99714 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6614234 0.93 HSD11B1 (0.46) HSD11B1CNR1MAPK1CCKBRHSD17B1
SCHEMBL6610827 0.90 HSD11B1 (0.52) HSD11B1SLC40A1CNR1CCKBRACLY
SCHEMBL6616741 0.88 HSD11B1 (0.66) HSD11B1CCKBRACLYALDH1A1
SCHEMBL6610632 0.84 HSD11B1 (0.46) HSD11B1CCKBRHPGD
SCHEMBL6624439 0.82 HSD11B1 (0.58) HSD11B1ACLYALDH1A1
SCHEMBL6628500 0.80 HSD11B1 (0.48) HSD11B1SLC40A1CNR1ITGAVCCKBR
SCHEMBL20899669 0.79 ACLY (0.44) HSD11B1SLC40A1ITGAVACLYALDH1A1
SCHEMBL3605392 0.79 HSD11B1 (0.80) HSD11B1HSD17B1HSD17B2
SCHEMBL6615038 0.79 HSD11B1 (0.57) HSD11B1SLC40A1MAPK1CCKBRHSD17B1
SCHEMBL6697889 0.78 HSD11B1 (0.54) HSD11B1ACLYALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004112779-A1 NEW USE VII BIOVITRUM AB (SE) 2004-12-29 WO claimed
EP-1461333-A1 INHIBITORS OF 11-BETA-HYDROXY STEROID DEHYDROGENASE TYPE 1 BIOVITRUM AB (SE) 2004-09-29 EP claimed
US-20030130279-A1 Inhibitors of 11-beta-hydroxy steroid dehydrogenase type 1 BIOVITRUM AB (SE) 2003-07-10 US claimed
WO-2003044009-A1 INHIBITORS OF 11-BETA-HYDROXY STEROID DEHYDROGENASE TYPE 1 BIOVITRUM AB (SE) 2003-05-30 WO claimed
EP-1461333-A1 INHIBITORS OF 11-BETA-HYDROXY STEROID DEHYDROGENASE TYPE 1 BIOVITRUM AB (SE) 2004-09-29 EP disclosed
US-20030130279-A1 Inhibitors of 11-beta-hydroxy steroid dehydrogenase type 1 BIOVITRUM AB (SE) 2003-07-10 US disclosed
WO-2003044009-A1 INHIBITORS OF 11-BETA-HYDROXY STEROID DEHYDROGENASE TYPE 1 BIOVITRUM AB (SE) 2003-05-30 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030130279-A1 Inhibitors of 11-beta-hydroxy steroid dehydrogenase type 1 HSD11B1, HSD17B1, HSD3B1 HSD11B1 1/4885SLC40A1 2287/4885CNR1 2499/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.