SCHEMBL6611036

SCHEMBL6611036

CCCN1C(=O)CNC(=O)C12CCN(CCc1ccccc1)CC2

nearest known ligand 0.58

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 10/20 0.52
LMNA P02545 1/20 0.49
CHRM2 P08172 1/20 0.49
ADRA2A P08913 1/20 0.49
CYP2D6 P10635 1/20 0.49
TSHR P16473 1/20 0.49
DRD1 P21728 1/20 0.49
MAPT P10636 1/20 0.48
KMT2A Q03164 1/20 0.48
CXCR3 P49682 1/20 0.48
SIGMAR1 Q99720 3/20 0.46
OPRM1 P35372 2/20 0.46
CXCR4 P61073 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6614177 0.93 CCR5 (0.57) CCR5CXCR3SIGMAR1CXCR4
SCHEMBL6612781 0.93 LMNA (0.53) LMNACHRM2ADRA2ACYP2D6TSHR
SCHEMBL6615208 0.92 CCR5 (0.61) CCR5CXCR3SIGMAR1OPRM1CXCR4
SCHEMBL6613900 0.91 CCR5 (0.63) CCR5CXCR3SIGMAR1CXCR4
SCHEMBL6611815 0.91 CCR5 (0.63) CCR5CXCR3SIGMAR1CXCR4
SCHEMBL6012726 0.89 CXCR3 (0.59) CCR5CXCR3OPRM1
SCHEMBL6612028 0.88 LMNA (0.51) CCR5LMNACHRM2ADRA2ACYP2D6
SCHEMBL6613037 0.87 SIGMAR1 (0.49) CCR5LMNACHRM2ADRA2ACYP2D6
SCHEMBL6612763 0.86 CCR5 (0.52) CCR5LMNACHRM2ADRA2ACYP2D6
SCHEMBL6613998 0.86 OPRL1 (0.56) CCR5LMNACHRM2ADRA2ACYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1236726-B1 TRIAZASPIRO 5.5]UNDECANE DERIVATIVES AND DRUGS CONTAINING THE SAME AS THE ACTIVE INGREDIENT ONO PHARMACEUTICAL CO (JP) 2004-12-01 EP disclosed
EP-1236726-A1 TRIAZASPIRO 5.5]UNDECANE DERIVATIVES AND DRUGS CONTAINING THE SAME AS THE ACTIVE INGREDIENT ONO PHARMACEUTICAL CO., LTD. (JP) 2002-09-04 EP disclosed