SCHEMBL6614945

SCHEMBL6614945

CNC(=O)Cc1sccc1NS(=O)(=O)c1cccc(Cl)c1C

nearest known ligand 0.46

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 13/20 0.46
HSD17B1 P14061 2/20 0.46
HSD17B2 P37059 2/20 0.46
SLC40A1 Q9NP59 1/20 0.45
EDNRB P24530 2/20 0.42
EDNRA P25101 2/20 0.42
ALDH1A1 P00352 1/20 0.41
GAA P10253 1/20 0.41
MAPT P10636 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
F2 P00734 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6615811 0.89 HSD11B1 (0.47) HSD11B1HSD17B1HSD17B2SLC40A1EDNRB
SCHEMBL6611468 0.89 HSD11B1 (0.48) HSD11B1HSD17B1HSD17B2SLC40A1EDNRB
SCHEMBL6613157 0.88 HSD11B1 (0.47) HSD11B1HSD17B1HSD17B2SLC40A1EDNRB
SCHEMBL6612682 0.86 HSD11B1 (0.50) HSD11B1HSD17B1HSD17B2SLC40A1EDNRB
SCHEMBL6611067 0.85 HSD11B1 (0.47) HSD11B1HSD17B1HSD17B2SLC40A1EDNRB
SCHEMBL6612479 0.84 HSD11B1 (0.48) HSD11B1HSD17B1HSD17B2SLC40A1EDNRB
SCHEMBL6692119 0.84 HSD11B1 (0.63) HSD11B1HSD17B1HSD17B2SLC40A1EDNRB
SCHEMBL6625131 0.83 HSD11B1 (0.52) HSD11B1HSD17B1HSD17B2SLC40A1EDNRB
SCHEMBL6614316 0.83 HSD11B1 (0.48) HSD11B1HSD17B1HSD17B2SLC40A1EDNRB
SCHEMBL6614921 0.83 SLC40A1 (0.47) HSD11B1HSD17B1HSD17B2SLC40A1EDNRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1461333-A1 INHIBITORS OF 11-BETA-HYDROXY STEROID DEHYDROGENASE TYPE 1 BIOVITRUM AB (SE) 2004-09-29 EP claimed
US-20030130279-A1 Inhibitors of 11-beta-hydroxy steroid dehydrogenase type 1 BIOVITRUM AB (SE) 2003-07-10 US claimed
WO-2003044009-A1 INHIBITORS OF 11-BETA-HYDROXY STEROID DEHYDROGENASE TYPE 1 BIOVITRUM AB (SE) 2003-05-30 WO claimed
WO-2019075394-A1 COMPOUNDS FOR TREATMENT OF EMOTIONAL/PSYCHOLOGICAL SYMPTOMS IN FRAGILE X SYNDROME VANDERKLISH PETER (US) 2019-04-18 WO disclosed
WO-2004112779-A1 NEW USE VII BIOVITRUM AB (SE) 2004-12-29 WO disclosed
EP-1461333-A1 INHIBITORS OF 11-BETA-HYDROXY STEROID DEHYDROGENASE TYPE 1 BIOVITRUM AB (SE) 2004-09-29 EP disclosed
US-20030130279-A1 Inhibitors of 11-beta-hydroxy steroid dehydrogenase type 1 BIOVITRUM AB (SE) 2003-07-10 US disclosed
WO-2003044009-A1 INHIBITORS OF 11-BETA-HYDROXY STEROID DEHYDROGENASE TYPE 1 BIOVITRUM AB (SE) 2003-05-30 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030130279-A1 Inhibitors of 11-beta-hydroxy steroid dehydrogenase type 1 HSD11B1, HSD17B1, HSD3B1 HSD11B1 1/4885HSD17B1 2/4885HSD17B2 6/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.