SCHEMBL6615697

SCHEMBL6615697

COc1cc2ccc(Br)c(C=O)c2cc1OC

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ERN1 O75460 5/20 0.54
PRKDC P78527 1/20 0.51
ALDH1A1 P00352 5/20 0.43
MAPT P10636 4/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
HPGD P15428 2/20 0.43
LMNA P02545 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
APAF1 O14727 1/20 0.42
TDP2 O95551 1/20 0.42
NSD2 O96028 1/20 0.42
CASP3 P42574 1/20 0.42
PPP1CA P62136 1/20 0.42
SENP8 Q96LD8 1/20 0.42
SENP7 Q9BQF6 1/20 0.42
SENP6 Q9GZR1 1/20 0.42
SAE1 Q9UBE0 1/20 0.42
UBA2 Q9UBT2 1/20 0.42
TSHR P16473 2/20 0.41
CYP3A4 P08684 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19305505 0.80 ERN1 (0.53) ERN1ALDH1A1MAPTHPGDSAE1
SCHEMBL8153548 0.79 ERN1 (0.45) ERN1ALDH1A1MAPTKDM4ERAD52
SCHEMBL6618916 0.78 PRKDC (0.41) ERN1PRKDCALDH1A1MAPTSAE1
SCHEMBL6618920 0.78 ALDH1A1 (0.42) ERN1PRKDCALDH1A1MAPTL3MBTL1
SCHEMBL28948932 0.76 TUBB4A (0.46) ERN1PRKDCALDH1A1MAPTHPGD
SCHEMBL19305517 0.76 IMPDH2 (0.45) PRKDCALDH1A1MAPTTSHRCYP3A4
SCHEMBL21122870 0.75 CYP2A6 (0.42) ERN1ALDH1A1MAPTSMN1; SMN2HPGD
SCHEMBL28118488 0.74 ALDH1A1 (0.45) ALDH1A1MAPTHPGDL3MBTL1APAF1
SCHEMBL16582712 0.74 SLC2A1 (0.44) ALDH1A1MAPTSMN1; SMN2HPGDL3MBTL1
SCHEMBL3268893 0.74 ERN1 (0.41) ERN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1042294-B1 HETEROCYCLIC CYTOTOXIC AGENTS UNIV RUTGERS (US) 2004-08-11 EP disclosed
US-6486167-B1 Heterocyclic cytotoxic agents RUTGERS, THE STATE UNIVERSITY OF NEW JERSEY 2002-11-26 US disclosed
CN-1286685-A Heterocyclic cytotoxic agents UNIV RUTGERS (US) 2001-03-07 CN disclosed
US-6140328-A FOR TREATING TUMOR RUTGERS, THE STATE UNIVERSITY OF NEW JERSEY (US) 2000-10-31 US disclosed
EP-1042294-A1 HETEROCYCLIC CYTOTOXIC AGENTS RUTGERS, THE STATE UNIVERSITY OF NEW JERSEY (US) 2000-10-11 EP disclosed
WO-1999031067-A1 HETEROCYCLIC CYTOTOXIC AGENTS RUTGERS, THE STATE UNIVERSITY OF NEW JERSEY (US) 1999-06-24 WO disclosed