SCHEMBL8153548

SCHEMBL8153548

COc1ccc2c(C=O)c(Br)ccc2c1

nearest known ligand 0.45

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ERN1 O75460 3/20 0.45
ALDH1A1 P00352 3/20 0.44
CYP1A2 P05177 1/20 0.43
CYP2A6 P11509 1/20 0.43
KDM4E B2RXH2 1/20 0.42
MAPT P10636 1/20 0.42
SLC2A1 P11166 2/20 0.41
MAPK1 P28482 1/20 0.40
RAD52 P43351 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30066982 0.82 MTNR1A (0.51) ERN1ALDH1A1CYP1A2CYP2A6MAPT
SCHEMBL10388887 0.82 MTNR1A (0.51) ERN1ALDH1A1CYP1A2CYP2A6MAPT
SCHEMBL18425254 0.82 ALDH1A1 (0.54) ERN1ALDH1A1CYP1A2CYP2A6KDM4E
SCHEMBL28948948 0.81 CYP1A2 (0.43) ERN1ALDH1A1CYP1A2CYP2A6KDM4E
SCHEMBL1360246 0.81 ERN1 (0.59) ERN1
SCHEMBL30066894 0.81 ERN1 (0.59) ERN1
SCHEMBL6615697 0.79 ERN1 (0.54) ERN1ALDH1A1KDM4EMAPTRAD52
SCHEMBL5660761 0.78 ALDH1A1 (0.46) ERN1ALDH1A1CYP1A2CYP2A6KDM4E
SCHEMBL27741565 0.77 CYP1A2 (0.52) ERN1ALDH1A1CYP1A2CYP2A6KDM4E
SCHEMBL19712480 0.77 ALDH1A1 (0.51) ALDH1A1CYP1A2KDM4EMAPTSLC2A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114573588-A Axial chiral benzopyrazine compound and preparation method and application thereof 中国科学院兰州化学物理研究所 2022-06-03 CN claimed
CN-114573588-A Axial chiral benzopyrazine compound and preparation method and application thereof 中国科学院兰州化学物理研究所 2022-06-03 CN disclosed
EP-1025074-A1 RECOVERY AND RECYCLE OF CATALYST COMPONENTS USED IN PALLADIUM-CATALYZED PREPARATION OF ARYLCARBOXYLIC ACIDS ALBEMARLE CORPORATION (US) 2000-08-09 EP disclosed
WO-1999019289-A1 RECOVERY AND RECYCLE OF CATALYST COMPONENTS USED IN PALLADIUM-CATALYZED PREPARATION OF ARYLCARBOXYLIC ACIDS ALBEMARLE CORPORATION (US) 1999-04-22 WO disclosed