SCHEMBL6617779

SCHEMBL6617779

CSC1C(=O)CCc2cc3c(cc21)OCO3

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 4/20 0.43
KDM4E B2RXH2 3/20 0.43
CASP1 P29466 3/20 0.43
ALDH1A1 P00352 2/20 0.43
GLA P06280 2/20 0.43
HPGD P15428 2/20 0.43
CASP7 P55210 2/20 0.43
HSD17B10 Q99714 2/20 0.43
GAA P10253 1/20 0.42
CYP3A4 P08684 4/20 0.41
HTR1A P08908 1/20 0.41
CHRNA7 P36544 3/20 0.40
ACHE P22303 1/20 0.40
DRD1 P21728 2/20 0.39
ADRA1A P35348 1/20 0.39
DRD2 P14416 1/20 0.39
CYP1A2 P05177 2/20 0.37
CYP2C9 P11712 2/20 0.37
TSHR P16473 2/20 0.37
CYP2C19 P33261 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8501452 0.72 CYP2D6 (0.35) CYP2D6KDM4ECASP1ALDH1A1GAA
SCHEMBL809535 0.70 KIF11 (0.41) CYP2D6KDM4ECASP1ALDH1A1GLA
SCHEMBL6615393 0.68 ACP3 (0.42)
SCHEMBL13343323 0.68 ALDH1A1 (0.53) KDM4ECASP1ALDH1A1HPGDHSD17B10
SCHEMBL13343320 0.67 MAPT (0.54) CYP2D6KDM4EALDH1A1HSD17B10CYP3A4
SCHEMBL9150060 0.62 KDM4E (0.54) CYP2D6KDM4ECASP1ALDH1A1GLA
SCHEMBL11006053 0.62 KDM4E (0.46) CYP2D6KDM4ECASP1ALDH1A1GLA
SCHEMBL12633798 0.62 MAOA (0.57) CYP2D6KDM4ECASP1ALDH1A1GLA
SCHEMBL6614937 0.61 KDM4E (0.44) CYP2D6KDM4ECASP1ALDH1A1GLA
SCHEMBL6336267 0.61 KDM4E (0.58) CYP2D6KDM4ECASP1CASP7HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1042294-B1 HETEROCYCLIC CYTOTOXIC AGENTS UNIV RUTGERS (US) 2004-08-11 EP disclosed
US-6486167-B1 Heterocyclic cytotoxic agents RUTGERS, THE STATE UNIVERSITY OF NEW JERSEY 2002-11-26 US disclosed
US-6140328-A FOR TREATING TUMOR RUTGERS, THE STATE UNIVERSITY OF NEW JERSEY (US) 2000-10-31 US disclosed