SCHEMBL6618503

SCHEMBL6618503

Nc1ccc2[nH]c(S(=O)(=O)c3ccccc3)cc2c1

nearest known ligand 0.54

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CA2 P00918 3/20 0.46
CYP2A6 P11509 1/20 0.45
KEAP1 Q14145 1/20 0.45
HTR6 P50406 4/20 0.41
LMNA P02545 2/20 0.41
AKR1B1 P15121 2/20 0.40
FFAR2 O15552 1/20 0.38
KDM4E B2RXH2 1/20 0.38
ALDH1A1 P00352 1/20 0.38
PARP1 P09874 1/20 0.37
CYP3A4 P08684 2/20 0.37
CYP2C9 P11712 2/20 0.37
MPO P05164 1/20 0.37
TSHR P16473 1/20 0.37
CNR1 P21554 1/20 0.37
CYP2C19 P33261 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3237494 0.82 CA2 (0.62) CA2CYP2A6HTR6LMNAAKR1B1
SCHEMBL31561597 0.82 CA2 (0.62) CA2CYP2A6HTR6LMNAAKR1B1
SCHEMBL7407839 0.81 CNR1 (0.54) CA2HTR6AKR1B1CNR1
SCHEMBL27867018 0.81 KDM4E (0.47) CA2HTR6LMNAAKR1B1KDM4E
SCHEMBL5190594 0.81 AKR1B1 (0.56) CA2HTR6LMNAAKR1B1FFAR2
SCHEMBL8120975 0.81 KDM4E (0.49) CA2HTR6KDM4ECYP3A4CYP2C9
SCHEMBL4629441 0.80 CA2 (0.57) CA2HTR6LMNAAKR1B1ALDH1A1
SCHEMBL19260939 0.79 KIF11 (0.43) CA2CYP2A6HTR6AKR1B1CNR1
SCHEMBL17803693 0.79 CA2 (0.42) CA2HTR6AKR1B1CNR1
SCHEMBL9561474 0.78 CYP19A1 (0.55) CA2HTR6LMNAAKR1B1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1444210-A1 QUNAZOLINE DERIVATIVES AS ANTITUMOR AGENTS AstraZeneca AB (SE) 2004-08-11 EP disclosed
WO-2003040108-A1 QUINAZOLINE DERIVATIVES AS ANTITUMOR AGENTS ASTRAZENECA AB (SE) 2003-05-15 WO disclosed