SCHEMBL6624341

SCHEMBL6624341

O=C(O)Nc1cc(OCC(F)(F)F)c(-c2ccccc2F)cc1NC(=O)CC(=O)c1cccc(-n2ccnn2)c1

nearest known ligand 0.37

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 1/20 0.36
SCN9A Q15858 1/20 0.35
POLB P06746 1/20 0.35
CYP3A4 P08684 1/20 0.35
TP53 P04637 1/20 0.34
MAPT P10636 1/20 0.34
RXFP1 Q9HBX9 1/20 0.34
ALDH1A1 P00352 2/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
UGCG Q16739 1/20 0.34
KEAP1 Q14145 1/20 0.34
SMN1; SMN2 Q16637 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6165283 0.90 NOTUM (0.34) NOTUMSCN9ACYP3A4TP53MAPT
SCHEMBL7704182 0.89 CYP3A4 (0.35) NOTUMCYP3A4TP53MAPTRXFP1
SCHEMBL7705397 0.82 KMT2A (0.40) NOTUMMAPTMEN1KMT2AKEAP1
SCHEMBL7139910 0.81 CYP3A4 (0.34) NOTUMCYP3A4ALDH1A1KEAP1SMN1; SMN2
SCHEMBL6610284 0.81 VCP (0.39) POLBUGCG
SCHEMBL7705335 0.78 ALDH1A1 (0.44) POLBCYP3A4TP53MAPTALDH1A1
SCHEMBL6167305 0.78 ABL1 (0.40) CYP3A4UGCG
SCHEMBL7704777 0.78 ALDH1A1 (0.39) CYP3A4TP53MAPTRXFP1ALDH1A1
SCHEMBL6622928 0.77 HSD11B1 (0.33) SCN9A
SCHEMBL7528469 0.77 KEAP1 (0.41) NOTUMCYP3A4MAPTALDH1A1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1379511-A1 DIHYDRO-BENZO (b) (1, 4) DIAZEPIN-2-ONE DERIVATIVES AS MGLUR2 ANTAGONISTS II F. HOFFMANN-LA ROCHE AG (CH) 2004-01-14 EP disclosed
WO-2002083652-A1 DIHYDRO-BENZO [b] [1, 4] DIAZEPIN-2-ONE DERIVATIVES AS MGLUR2 ANTAGONISTS II F. HOFFMANN-LA ROCHE AG (CH) 2002-10-24 WO disclosed