SCHEMBL6626285

SCHEMBL6626285

CC(C(=O)O)N1CCN(C(CO)C(=O)O)CCN(CC(=O)O)CCN(C(CO)C(=O)O)CC1

nearest known ligand 0.47

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
SLC6A9 P48067 1/20 0.39
HSD17B10 Q99714 1/20 0.36
TACR1 P25103 3/20 0.35
SIGMAR1 Q99720 1/20 0.34
KDM4E B2RXH2 1/20 0.33
MME P08473 1/20 0.33
ALB P02768 1/20 0.32
ALDH1A1 P00352 2/20 0.32
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32
S1PR1 P21453 1/20 0.30
NPC1 O15118 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6628233 0.94 SLC6A9 (0.36) SLC6A9HSD17B10TACR1SIGMAR1KDM4E
SCHEMBL5551081 0.90 SLC6A9 (0.45) SLC6A9HSD17B10TACR1ALBMEN1
SCHEMBL6628577 0.90 SLC6A9 (0.45) SLC6A9HSD17B10TACR1ALBMEN1
SCHEMBL6625142 0.90 SLC6A9 (0.45) SLC6A9HSD17B10TACR1ALBMEN1
SCHEMBL5370149 0.90 SLC6A9 (0.45) SLC6A9HSD17B10TACR1ALBMEN1
SCHEMBL7590528 0.88 SLC6A9 (0.46) SLC6A9HSD17B10TACR1SIGMAR1KDM4E
SCHEMBL13223371 0.88 SLC6A9 (0.46) SLC6A9HSD17B10TACR1SIGMAR1KDM4E
SCHEMBL5033230 0.88 SLC6A9 (0.46) SLC6A9HSD17B10TACR1SIGMAR1KDM4E
SCHEMBL16582365 0.88 SLC6A9 (0.46) SLC6A9HSD17B10TACR1SIGMAR1KDM4E
SCHEMBL16382945 0.88 SLC6A9 (0.46) SLC6A9HSD17B10TACR1SIGMAR1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0998476-B1 1,4,7,10-TETRAAZABICYCLO 8.2.2]TETRADECAN-2-ONE, A PROCESS FOR THE PREPARATION THEREOF AND THE USE THEREOF FOR THE PREPARATION OF TETRAAZAMACROCYCLES BRACCO SPA (IT) 2004-05-06 EP disclosed
US-6162912-A Process of preparing tetraacetic acid derivatives DIBRA S.P.A. (IT) 2000-12-19 US disclosed
US-6028194-A SYNTHESIS OF GADOTERIDOL AND GADOBUTROL CONTRAST AGENTS FOR THE RESONANCE TECHNIQUE (MAGNETIC RESONANCE IMAGING) DIBRA S.P.A. (IT) 2000-02-22 US disclosed
US-6020485-A Process for producing tetraazabicyclo monoacetic acid DIBRA S.P.A. (IT) 2000-02-01 US disclosed
US-5977353-A 1,4,7,10-tetraazabicyclo[8.2.2]tetradecan-2-one, a process for the preparation thereof and the use thereof for the preparation of tetraazamacrocycles DIBRA S.P.A. (IT) 1999-11-02 US disclosed