SCHEMBL6628577

SCHEMBL6628577

O=C(O)CN1CCN(C(CO)C(=O)O)CCN(C(CO)C(=O)O)CCN(C(CO)C(=O)O)CC1

nearest known ligand 0.58

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
SLC6A9 P48067 1/20 0.45
HSD17B10 Q99714 1/20 0.42
ALB P02768 1/20 0.35
TACR1 P25103 3/20 0.34
CACNA2D1 P54289 2/20 0.33
CACNA1B Q00975 2/20 0.33
CACNB1 Q02641 2/20 0.33
CACNA1C Q13936 2/20 0.33
LMNA P02545 1/20 0.33
S1PR1 P21453 1/20 0.31
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6625142 1.00 SLC6A9 (0.45) SLC6A9HSD17B10ALBTACR1CACNA2D1
SCHEMBL5370149 1.00 SLC6A9 (0.45) SLC6A9HSD17B10ALBTACR1CACNA2D1
SCHEMBL5551081 1.00 SLC6A9 (0.45) SLC6A9HSD17B10ALBTACR1CACNA2D1
SCHEMBL6626285 0.90 SLC6A9 (0.39) SLC6A9HSD17B10ALBTACR1S1PR1
SCHEMBL21185731 0.87 SLC6A9 (0.44) SLC6A9HSD17B10ALBTACR1CACNA2D1
SCHEMBL300399 0.85
SCHEMBL9159811 0.85 SLC6A9 (0.43) SLC6A9HSD17B10ALBTACR1CACNA2D1
SCHEMBL6628233 0.85 SLC6A9 (0.36) SLC6A9HSD17B10ALBTACR1S1PR1
SCHEMBL15780321 0.85 SLC6A9 (0.45) SLC6A9HSD17B10ALBTACR1
SCHEMBL2779265 0.85 SLC6A9 (0.45) SLC6A9HSD17B10ALBTACR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0325762-B1 Macrocyclic chelating agents and chelates thereof BRACCO SPA (IT) 1995-03-22 EP claimed
EP-0325762-A1 Macrocyclic chelating agents and chelates thereof BRACCO S.p.A. (IT) 1989-08-02 EP claimed
EP-0998476-B1 1,4,7,10-TETRAAZABICYCLO 8.2.2]TETRADECAN-2-ONE, A PROCESS FOR THE PREPARATION THEREOF AND THE USE THEREOF FOR THE PREPARATION OF TETRAAZAMACROCYCLES BRACCO SPA (IT) 2004-05-06 EP disclosed
US-6162912-A Process of preparing tetraacetic acid derivatives DIBRA S.P.A. (IT) 2000-12-19 US disclosed
US-6048980-A AMINATION WITH DEHYDROHALOGENATION FOLLOWED BY HYDROLYSIS OF ESTER GROUP DIBRA S.P.A (IT) 2000-04-11 US disclosed
US-6028194-A SYNTHESIS OF GADOTERIDOL AND GADOBUTROL CONTRAST AGENTS FOR THE RESONANCE TECHNIQUE (MAGNETIC RESONANCE IMAGING) DIBRA S.P.A. (IT) 2000-02-22 US disclosed
US-6020485-A Process for producing tetraazabicyclo monoacetic acid DIBRA S.P.A. (IT) 2000-02-01 US disclosed
US-5977353-A 1,4,7,10-tetraazabicyclo[8.2.2]tetradecan-2-one, a process for the preparation thereof and the use thereof for the preparation of tetraazamacrocycles DIBRA S.P.A. (IT) 1999-11-02 US disclosed
EP-0325762-B1 Macrocyclic chelating agents and chelates thereof BRACCO SPA (IT) 1995-03-22 EP disclosed
US-5132409-A Derivatives of 1,4,7,10-Tetraazacyclododecane BRACCO INDUSTRIA CHIMICA S.P.A. (IT) 1992-07-21 US disclosed
EP-0325762-A1 Macrocyclic chelating agents and chelates thereof BRACCO S.p.A. (IT) 1989-08-02 EP disclosed