SCHEMBL6627151

SCHEMBL6627151

Cc1ccc(C)c(C=O)n1

nearest known ligand 0.39

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.39
CCR1 P32246 3/20 0.39
RAB9A P51151 1/20 0.39
CCR5 P51681 1/20 0.39
S100A4 P26447 1/20 0.38
OPRK1 P41145 1/20 0.36
KMT2A Q03164 1/20 0.36
TSHR P16473 1/20 0.34
CYP1A2 P05177 4/20 0.33
HTR2B P41595 1/20 0.33
CCR8 P51685 1/20 0.32
CYP2A6 P11509 1/20 0.32
KDM4C Q9H3R0 1/20 0.31
NOS2 P35228 3/20 0.31
NOS1 P29475 2/20 0.31
ADORA2A P29274 1/20 0.31
ADORA1 P30542 1/20 0.31
KDM4E B2RXH2 1/20 0.30
NOS3 P29474 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15927725 0.79 CCR1 (0.37) ALDH1A1CCR1RAB9ACCR5S100A4
SCHEMBL18150327 0.77 CCR1 (0.41) ALDH1A1CCR1RAB9ACCR5S100A4
SCHEMBL1390456 0.77 KDM4E (0.45) ALDH1A1CCR1RAB9ACCR5S100A4
SCHEMBL29792042 0.77 TGFBR1 (0.38) ALDH1A1CCR1RAB9ACCR5S100A4
SCHEMBL17429949 0.77 TGFBR1 (0.38) ALDH1A1CCR1RAB9ACCR5S100A4
SCHEMBL23641383 0.77 CCR1 (0.36) ALDH1A1CCR1RAB9ACCR5S100A4
SCHEMBL2226680 0.77 CYP3A4 (0.35) ALDH1A1KMT2ATSHRCYP1A2HTR2B
SCHEMBL22342564 0.77 ALDH1A1 (0.32) ALDH1A1TSHRHTR2BCYP2A6
SCHEMBL29952500 0.77 CYP3A4 (0.35) ALDH1A1KMT2ATSHRCYP1A2HTR2B
SCHEMBL31337139 0.77 ALDH1A1 (0.32) ALDH1A1TSHRHTR2BCYP2A6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20170174654-A1 COMPOUNDS AND USES THEREOF FOR THE MODULATION OF HEMOGLOBIN GLOBAL BLOOD THERAPEUTICS, INC. 2017-06-22 US disclosed
US-9422279-B2 Compounds and uses thereof for the modulation of hemoglobin GLOBAL BLOOD THERAPEUTICS, INC. (US) 2016-08-23 US disclosed
US-20160193191-A1 ANTAGONISTS OF CHEMOKINE RECEPTORS CHEMOCENTRYX, INC. 2016-07-07 US disclosed
US-9181241-B2 Antagonists of chemokine receptors CHEMOCENTRYX, INC. (US) 2015-11-10 US disclosed
US-20140275152-A1 Compounds and uses thereof for the modulation of hemoglobin GLOBAL BLOOD THERAPEUTICS, INC. 2014-09-18 US disclosed
US-20140057937-A1 ANTAGONISTS OF CHEMOKINE RECEPTORS CHEMOCENTRYX, INC. (US) 2014-02-27 US disclosed
EP-0974602-B1 Catalyst and process for hydrogenating olefinically unsaturated compound JSR CORP (JP) 2004-01-02 EP disclosed
US-6291596-B1 CONTACTING OLEFINICALLY UNSATURATED COMPOUND WITH HYDROGEN IN THE PRESENCE OF A HYDROGENATION CATALYST COMPRISING TITANIUM OR ZIRCONIUM OR HAFNIUM COMPOUND IN AN INERT, ORGANIC SOLVENT JSR CORPORATION (JP) 2001-09-18 US disclosed
EP-0974602-A1 Catalyst and process for hydrogenating olefinically unsaturated compound JSR Corporation (JP) 2000-01-26 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20170174654-A1 COMPOUNDS AND USES THEREOF FOR THE MODULATION OF HEMOGLOBIN HBG2, HBG1, HBB ALDH1A1 1089/4885CCR1 3836/4885RAB9A 3417/4885
US-20160193191-A1 ANTAGONISTS OF CHEMOKINE RECEPTORS CCR1, CCR3, CCR2 ALDH1A1 1354/4885CCR1 1/4885RAB9A 3905/4885
US-20140275152-A1 Compounds and uses thereof for the modulation of hemoglobin HBG2, HBG1, HBB ALDH1A1 1089/4885CCR1 3836/4885RAB9A 3417/4885
US-20140057937-A1 ANTAGONISTS OF CHEMOKINE RECEPTORS CCR1, CCR3, CCR2 ALDH1A1 1354/4885CCR1 1/4885RAB9A 3905/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.