SCHEMBL6629448

SCHEMBL6629448

NC(=O)c1ccccc1Sc1cccs1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIRT1 Q96EB6 1/20 0.57
ALDH1A1 P00352 5/20 0.40
MAPT P10636 4/20 0.40
KDM4E B2RXH2 4/20 0.40
HSD17B10 Q99714 3/20 0.40
HPGD P15428 2/20 0.40
TSHR P16473 2/20 0.40
NPC1 O15118 2/20 0.40
TP53 P04637 2/20 0.40
RAB9A P51151 2/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
GAA P10253 2/20 0.40
NFKB1 P19838 1/20 0.40
NFKB2 Q00653 1/20 0.40
RELA Q04206 1/20 0.40
FBP1 P09467 1/20 0.39
PDE7A Q13946 2/20 0.38
MAPK1 P28482 2/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27274014 0.83 FBP1 (0.39) SIRT1ALDH1A1MAPTKDM4ENPC1
SCHEMBL3077375 0.80 SIRT1 (0.77) SIRT1ALDH1A1MAPTKDM4EHSD17B10
SCHEMBL6633843 0.76 SIRT1 (0.53) SIRT1ALDH1A1MAPTKDM4EHSD17B10
SCHEMBL7701766 0.74 SIRT1 (0.54) SIRT1ALDH1A1MAPTKDM4EHSD17B10
SCHEMBL6633964 0.74 SIRT1 (0.54) SIRT1ALDH1A1MAPTKDM4EHSD17B10
SCHEMBL1030659 0.73 SIRT1 (1.00) SIRT1ALDH1A1MAPTKDM4EHSD17B10
SCHEMBL11821622 0.72 SIRT1 (0.64) SIRT1ALDH1A1MAPTKDM4EHSD17B10
SCHEMBL29530768 0.72 SIRT1 (0.64) SIRT1ALDH1A1MAPTKDM4EHSD17B10
SCHEMBL1399456 0.72 SIRT1 (0.64) SIRT1ALDH1A1MAPTKDM4EHSD17B10
SCHEMBL6629741 0.72 SIRT1 (0.65) SIRT1ALDH1A1MAPTKDM4EHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1480977-A2 SUBSTITUTED ARYL COMPOUNDS FOR TREATMENT OF DISEASE PHARMACIA & UPJOHN COMPANY (US) 2004-12-01 EP claimed
WO-2003070728-A2 AZABICYCLO-SUBSTITUTED BENZOYLAMIDES AND THIOAMIDES FOR TREATMENT OF CNS-RELATED DISORDERS PHARMACIA & UPJOHN COMPANY (US) 2003-08-28 WO claimed
WO-2002016357-A2 QUINUCLIDINE-SUBSTITUTED ARYL MOIETIES FOR TREATMENT OF DISEASE (NICOTINIC ACETYLCHOLINE RECEPTOR LIGANDS) PHARMACIA & UPJOHN COMPANY (US) 2002-02-28 WO claimed